SCHEMBL3264576

SCHEMBL3264576

COC(=O)C(Br)CN(CC(=O)OC(C)(C)C)CC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ZDHHC7 Q9NXF8 1/20 0.40
CA12 O43570 3/20 0.33
CA14 Q9ULX7 3/20 0.33
CYP2D6 P10635 1/20 0.32
DGAT1 O75907 1/20 0.32
NR1D1 P20393 2/20 0.31
CA2 P00918 2/20 0.30
CA1 P00915 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3780438 0.80 CYP2D6 (0.35) CYP2D6NR1D1CA2CA1
SCHEMBL15952123 0.78 CYP2D6 (0.42) ZDHHC7CA12CA14CYP2D6DGAT1
SCHEMBL15952124 0.78 CYP2D6 (0.42) ZDHHC7CA12CA14CYP2D6DGAT1
SCHEMBL9338982 0.75 CYP2D6 (0.37) CYP2D6NR1D1CA2CA1
SCHEMBL14729341 0.75 CA12 (0.41) CA12CA14CYP2D6DGAT1NR1D1
SCHEMBL13965219 0.75 CA12 (0.41) CA12CA14CYP2D6DGAT1NR1D1
SCHEMBL17754726 0.75 ZDHHC7 (0.47) ZDHHC7CA12CA14CYP2D6DGAT1
SCHEMBL22737498 0.74 CYP2D6 (0.35) CA12CA14CYP2D6DGAT1NR1D1
SCHEMBL3780442 0.74 TDP1 (0.32) CYP2D6NR1D1
SCHEMBL27420033 0.74 NR1D1 (0.38) CA12CA14CYP2D6DGAT1NR1D1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010011367-A2 BIMODAL LIGANDS WITH MACROCYCLIC AND ACYCLIC BINDING MOIETIES, COMPLEXES AND COMPOSITIONS THEREOF, AND METHODS OF USING ILLINOIS INSTITUTE OF TECHNOLOGY (US) 2010-01-28 WO disclosed