SCHEMBL3265228

SCHEMBL3265228

CN(C)CCOc1cccc(CN(CCO)C(=O)c2nc3ccc(-c4ccnc(N)n4)cc3s2)c1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 10/20 0.58
ROCK1 Q13464 3/20 0.58
CDC42BPA Q5VT25 2/20 0.58
MAPK10 P53779 1/20 0.58
CYP3A4 P08684 1/20 0.42
PIK3CA P42336 7/20 0.41
HDAC1 Q13547 1/20 0.40
MTOR P42345 1/20 0.37
PFKFB3 Q16875 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13457310 0.89 ROCK2 (0.72) ROCK2ROCK1CDC42BPAMAPK10CYP3A4
SCHEMBL3241319 0.88 ROCK2 (0.56) ROCK2ROCK1CDC42BPAMAPK10CYP3A4
SCHEMBL13457103 0.85 ROCK2 (0.71) ROCK2ROCK1CDC42BPAMAPK10PIK3CA
SCHEMBL3265194 0.85 ROCK2 (0.78) ROCK2ROCK1CDC42BPAMAPK10CYP3A4
SCHEMBL3265491 0.84 ROCK2 (0.54) ROCK2ROCK1CDC42BPAMAPK10CYP3A4
SCHEMBL13457234 0.82 ROCK2 (0.53) ROCK2ROCK1CDC42BPAMAPK10CYP3A4
SCHEMBL3264837 0.80 ROCK2 (0.56) ROCK2ROCK1CDC42BPAMAPK10
SCHEMBL13457417 0.78 ROCK2 (0.48) ROCK2ROCK1CDC42BPAMAPK10PIK3CA
SCHEMBL3261889 0.78 ROCK2 (0.71) ROCK2ROCK1CDC42BPAMAPK10CYP3A4
SCHEMBL3262928 0.76 ROCK2 (0.68) ROCK2ROCK1CDC42BPAMAPK10CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010024903-A1 BENZO[d]OXAZOLES AND BENZO[d]THIAZOLES AS KINASE INHIBITORS FENG YANGBO (US) 2010-03-04 WO disclosed
WO-2010024903-A1 BENZO[d]OXAZOLES AND BENZO[d]THIAZOLES AS KINASE INHIBITORS FENG YANGBO (US) 2010-03-04 WO disclosed