SCHEMBL3265533

SCHEMBL3265533

COC(c1ccccc1)N1CCCc2ccccc2C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 7/20 0.44
DRD5 P21918 6/20 0.40
DRD2 P14416 4/20 0.40
DRD4 P21917 4/20 0.40
DRD3 P35462 4/20 0.40
NPSR1 Q6W5P4 2/20 0.40
LMNA P02545 2/20 0.40
CYP1A2 P05177 4/20 0.40
CYP3A4 P08684 4/20 0.40
CYP2D6 P10635 4/20 0.40
CYP2C9 P11712 4/20 0.40
KCNA5 P22460 4/20 0.40
CYP2C19 P33261 4/20 0.40
KCNH2 Q12809 4/20 0.40
MAOA P21397 2/20 0.40
MAOB P27338 2/20 0.40
RIPK1 Q13546 2/20 0.39
TSHR P16473 1/20 0.39
KCNE1 P15382 1/20 0.39
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20536090 0.76 CYP2D6 (0.54) DRD1DRD3LMNACYP1A2CYP3A4
SCHEMBL11530901 0.76 CYP2D6 (0.36) DRD1DRD3NPSR1LMNACYP1A2
SCHEMBL12533128 0.75 HRH3 (0.50) DRD1DRD5LMNACYP2D6KCNH2
SCHEMBL4392254 0.73 CYP2D6 (0.45) DRD1DRD3LMNACYP1A2CYP3A4
SCHEMBL5213186 0.73 LMNA (0.64) NPSR1LMNARIPK1TSHRMEN1
SCHEMBL6184552 0.72 CYP2D6 (0.42) DRD1DRD3LMNACYP1A2CYP3A4
SCHEMBL28041845 0.71 CYP2D6 (0.40) DRD1DRD3LMNACYP1A2CYP3A4
SCHEMBL8480869 0.70 MAPK1 (0.45) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL10527232 0.69 MEN1 (0.59) CYP3A4CYP2D6KCNH2MEN1KMT2A
SCHEMBL5221988 0.69 CHRM2 (0.50) LMNACYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010012812-A1 BENZAZEPINES AND BENZAZOCINES AS SIGMA-RECEPTOR LIGANDES Westfälische Wilhelms Universität Münster (DE) 2010-02-04 WO disclosed