SCHEMBL11530901

SCHEMBL11530901

COC(c1ccccc1)N1CCC2=C(CCCC2)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 6/20 0.36
KCNH2 Q12809 5/20 0.36
CYP1A2 P05177 4/20 0.36
CYP3A4 P08684 4/20 0.36
CYP2C9 P11712 4/20 0.36
KCNA5 P22460 4/20 0.36
CYP2C19 P33261 4/20 0.36
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
KCNE1 P15382 1/20 0.35
OPRM1 P35372 3/20 0.33
CHRM2 P08172 2/20 0.33
CHRM4 P08173 2/20 0.33
CHRM5 P08912 2/20 0.33
CHRM1 P11229 2/20 0.33
CHRM3 P20309 2/20 0.33
OPRD1 P41143 2/20 0.33
OPRK1 P41145 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20536090 0.76 CYP2D6 (0.54) CYP2D6KCNH2CYP1A2CYP3A4CYP2C9
SCHEMBL3265533 0.76 DRD1 (0.44) CYP2D6KCNH2CYP1A2CYP3A4CYP2C9
SCHEMBL4392254 0.73 CYP2D6 (0.45) CYP2D6KCNH2CYP1A2CYP3A4CYP2C9
SCHEMBL10527232 0.69 MEN1 (0.59) CYP2D6KCNH2CYP3A4MEN1KMT2A
SCHEMBL6184552 0.69 CYP2D6 (0.42) CYP2D6KCNH2CYP1A2CYP3A4CYP2C9
SCHEMBL8480869 0.67 MAPK1 (0.45) CYP2D6KCNH2CYP1A2CYP3A4CYP2C9
SCHEMBL17513224 0.66 CYP2D6 (0.39) CYP2D6KCNH2CYP1A2CYP3A4CYP2C9
SCHEMBL5221988 0.66 CHRM2 (0.50) CYP2D6CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL7209211 0.65 L3MBTL1 (0.46) CYP3A4CYP2C19ALDH1A1MEN1KMT2A
SCHEMBL1845086 0.59 KMT2A (0.46) CYP2D6KCNH2CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4139534-A Process for the preparation of 14-hydroxymorphinan derivatives BRISTOL-MYERS COMPANY (US) 1979-02-13 US disclosed