SCHEMBL326797

SCHEMBL326797

COc1ccc(-c2nc(-c3ccc(OC)c(OC)c3)c3ccccc3n2)cc1F

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 15/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
ABCB1 P08183 9/20 0.56
ABCC1 P33527 5/20 0.56
WHR1 P49842 1/20 0.54
TP53 P04637 1/20 0.53
MAPT P10636 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
ACACA Q13085 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25082162 0.84 ABCG2 (0.58) ABCG2ABCB1ABCC1WHR1TP53
SCHEMBL8816999 0.83 ABCG2 (0.47) ABCG2L3MBTL1ABCB1ABCC1WHR1
SCHEMBL6001414 0.82 ABCG2 (0.58) ABCG2L3MBTL1ABCB1ABCC1WHR1
SCHEMBL8818335 0.79 L3MBTL1 (0.53) ABCG2L3MBTL1ABCB1ABCC1WHR1
SCHEMBL28054620 0.78 ABCG2 (0.65) ABCG2L3MBTL1ABCB1ABCC1TP53
SCHEMBL8779739 0.78 ABCG2 (0.49) ABCG2L3MBTL1ABCB1ABCC1TP53
SCHEMBL8779566 0.77 ABCG2 (0.48) ABCG2L3MBTL1ABCB1ABCC1TP53
SCHEMBL3786521 0.76 ABCG2 (0.47) ABCG2L3MBTL1ABCB1ABCC1TP53
SCHEMBL182874 0.76 PDGFRB (0.48) L3MBTL1SMN1; SMN2
SCHEMBL27767946 0.75 L3MBTL1 (0.58) ABCG2L3MBTL1ABCB1ABCC1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049502-B1 2,4-SUBSTITUTED QUINAZOLINES AS LIPID KINASE INHIBITORS NOVARTIS AG (CH) 2012-01-04 EP claimed