SCHEMBL3268115

SCHEMBL3268115

Cc1cc(Nc2cc(N3CCCC(NC(=O)c4cc5ccccc5s4)C3)nc3ccnn23)nn1C

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.45
DPP4 P27487 13/20 0.45
CHRNA7 P36544 4/20 0.38
HTR3A P46098 3/20 0.38
HTR1A P08908 1/20 0.38
DRD2 P14416 1/20 0.38
HTR2A P28223 1/20 0.38
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3268106 1.00 BTK (0.45) BTKDPP4CHRNA7HTR3AHTR1A
SCHEMBL3260799 0.87 BTK (0.47) BTKDPP4CHRNA7HTR3AHTR3E
SCHEMBL3262494 0.84 BTK (0.46) BTKDPP4CHRNA7HTR3AHTR1A
SCHEMBL2490136 0.82 BTK (0.46) BTKCHRNA7HTR3AHTR1ADRD2
SCHEMBL2493885 0.82 BTK (0.46) BTKCHRNA7HTR3AHTR1ADRD2
SCHEMBL3263368 0.76 DPP4 (0.40) BTKDPP4
SCHEMBL3263367 0.76 DPP4 (0.40) BTKDPP4
SCHEMBL13303488 0.74 DPP4 (0.54) DPP4
SCHEMBL19971540 0.74 BTK (0.40) BTKCHRNA7HTR3AHTR1ADRD2
SCHEMBL9984552 0.72 BTK (0.44) BTKCHRNA7HTR3AHTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010068806-A1 AMIDE DERIVATIVES AS BTK INHIBITORS IN THE TREATMENT OF ALLERGIC, AUTOIMMUNE AND INFLAMMATORY DISORDERS AS WELL AS CANCER CGI PHARMACEUTICALS, INC. (US) 2010-06-17 WO claimed