SCHEMBL3268262

SCHEMBL3268262

Cc1cccc(Sc2c(OC(N)=O)[nH]c3sccc23)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ICAM1 P05362 2/20 0.38
SELE P16581 2/20 0.38
MAPK8 P45983 1/20 0.33
KDR P35968 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
PARP15 Q460N3 3/20 0.32
TNKS2 Q9H2K2 3/20 0.32
PARP10 Q53GL7 2/20 0.32
PARP2 Q9UGN5 2/20 0.32
PARP14 Q460N5 1/20 0.32
TNKS O95271 1/20 0.32
PARP1 P09874 1/20 0.32
GCK P35557 1/20 0.32
TUBB4A P04350 2/20 0.32
TUBB P07437 2/20 0.32
TUBA3C P0DPH7 2/20 0.32
TUBA1B P68363 2/20 0.32
TUBA4A P68366 2/20 0.32
TUBB4B P68371 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3268815 0.88 TNKS2 (0.38) MAPK8MEN1KMT2APARP15TNKS2
SCHEMBL3275192 0.87 EDNRA (0.46) MAPK8MEN1KMT2APARP15TNKS2
SCHEMBL3269919 0.87 PDE4B (0.38) MAPK8MEN1KMT2APARP15TNKS2
SCHEMBL3270312 0.86 TNKS2 (0.39) MEN1KMT2APARP15TNKS2PARP10
SCHEMBL3177241 0.83 ICAM1 (0.42) ICAM1SELEMAPK8KDRPARP15
SCHEMBL3268577 0.82 KDR (0.39) ICAM1SELEMAPK8KDRPARP1
SCHEMBL3269142 0.81 PARP15 (0.33) PARP15TNKS2PARP10PARP2PARP14
SCHEMBL3268792 0.79 CDC7 (0.36) PARP15TNKS2PARP10PARP2TNKS
SCHEMBL3268877 0.78 PARP15 (0.35) MEN1KMT2APARP15TNKS2PARP10
SCHEMBL3270015 0.76 TUBB4A (0.42) MAPK8PARP15TNKS2PARP10PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784409-B1 SUBSTITUTED THIENOPYRROLE CARBOXYLIC ACID AMIDES, PYRROLOTHIAZOLE CARBOXYLIC ACID AMIDES, AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON AVENTIS PHARMA INC (US) 2010-06-16 EP claimed