SCHEMBL3273689

SCHEMBL3273689

COC(=O)c1[nH]c(O[Si](C)(C)C(C)(C)C)cc1C

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 5/20 0.35
RAF1 P04049 1/20 0.35
MAPT P10636 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
XDH P47989 1/20 0.33
CSNK2A2 P19784 1/20 0.33
KDR P35968 1/20 0.33
CSNK2B P67870 1/20 0.33
CSNK2A1 P68400 1/20 0.33
CYP3A4 P08684 1/20 0.32
ACHE P22303 1/20 0.32
MAPK1 P28482 1/20 0.32
CYP1A2 P05177 1/20 0.32
ATM Q13315 1/20 0.32
KDM4C Q9H3R0 1/20 0.32
DRD2 P14416 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13382878 0.74 AR (0.34) MAPT
SCHEMBL13382786 0.71 ALDH1A1 (0.45) MAPTMAPK1ALDH1A1LMNA
SCHEMBL23923776 0.71 ALDH1A1 (0.43) MAPK14RAF1MAPTXDHCYP3A4
SCHEMBL22397177 0.70 KDM4C (0.41) MAPTRAB9ACSNK2A2KDRCSNK2B
SCHEMBL28618724 0.70 CYP1A2 (0.52) MAPTRAB9AXDHCYP3A4ACHE
SCHEMBL2201771 0.69 CA12 (0.43) MAPTNPC1RAB9AKDRCYP3A4
SCHEMBL7517428 0.69 NOTUM (0.55) MAPTNPC1RAB9AXDHATM
SCHEMBL20046200 0.69 CA1 (0.43) MAPTNPC1RAB9ACYP1A2ATM
SCHEMBL30007012 0.69 CA12 (0.43) MAPTNPC1RAB9AKDRCYP3A4
SCHEMBL3023269 0.68 KDM4E (0.50) MAPTNPC1RAB9ACYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7691896-B2 Analogs of salinosporamide A PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-04-06 US disclosed
US-7691896-B2 Analogs of salinosporamide A PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-04-06 US disclosed
EP-1931679-A4 ANALOGS OF SALINOSPORAMIDE A HARVARD COLLEGE (US) 2009-07-29 EP disclosed
US-20090054665-A1 ANALOGS OF SALINOSPORAMIDE A PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2009-02-26 US disclosed
US-20090054665-A1 ANALOGS OF SALINOSPORAMIDE A PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2009-02-26 US disclosed
EP-1931679-A1 ANALOGS OF SALINOSPORAMIDE A The President and Fellows of Harvard College (US) 2008-06-18 EP disclosed
WO-2007021897-A1 ANALOGS OF SALINOSPORAMIDE A PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2007-02-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090054665-A1 ANALOGS OF SALINOSPORAMIDE A PSME1, PSMG3, PSMD5 MAPK14 2060/4885RAF1 1851/4885MAPT 3047/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.