Oleamide

Oleamide

SCHEMBL3280975

CCCCCCCC/C=C\CCCCCCCC(N)=O.O=C(O)/C=C\C(=O)O

nearest known ligand 0.82

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2BTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3MPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PPARGSLC6A2SLC6A3SLC6A4SMOTYK2pol

The experimentally established mechanism targets of Oleamide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG known ✓ P37231 3/20 0.65
SLC6A2 known ✓ P23975 1/20 0.65
SOAT1 P35610 2/20 0.82
FAAH O00519 2/20 0.82
CYP1A2 P05177 2/20 0.82
CYP2C19 P33261 2/20 0.82
KMT2A Q03164 2/20 0.82
MEN1 O00255 1/20 0.82
TP53 P04637 1/20 0.82
CYP3A4 P08684 1/20 0.82
KDM4E B2RXH2 2/20 0.74
CNR1 P21554 1/20 0.66
TERT O14746 3/20 0.65
PTPN1 P18031 3/20 0.65
PPARD Q03181 3/20 0.65
PPARA Q07869 3/20 0.65
MAPT P10636 2/20 0.65
BLM P54132 2/20 0.65
HSD17B10 Q99714 2/20 0.65
FABP4 P15090 2/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Maleic Acid SCHEMBL3281709 1.00 SOAT1 (0.82) SOAT1FAAHCYP1A2CYP2C19KMT2A
Oleamide SCHEMBL22285887 0.93 FAAH (0.96) SOAT1FAAHCYP1A2CYP2C19KMT2A
Oleamide SCHEMBL19814150 0.91 FAAH (1.00) SOAT1FAAHCYP1A2CYP2C19KMT2A
SCHEMBL21501560 0.91 FAAH (1.00) SOAT1FAAHCYP1A2CYP2C19KMT2A
SCHEMBL3228539 0.91 FAAH (1.00) SOAT1FAAHCYP1A2CYP2C19KMT2A
SCHEMBL24340776 0.91 FAAH (1.00) SOAT1FAAHCYP1A2CYP2C19KMT2A
SCHEMBL21983255 0.91 FAAH (1.00) SOAT1FAAHCYP1A2CYP2C19KMT2A
SCHEMBL22419041 0.91 FAAH (1.00) SOAT1FAAHCYP1A2CYP2C19KMT2A
SCHEMBL23528231 0.91 FAAH (1.00) SOAT1FAAHCYP1A2CYP2C19KMT2A
SCHEMBL21654359 0.91 FAAH (1.00) SOAT1FAAHCYP1A2CYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150072905-A1 VISCOELASTIC COMPOSITIONS SCHLUMBERGER TECHNOLOGY CORP (US) 2015-03-12 US disclosed
US-7704926-B2 Viscoelastic compositions SCHLUMBERGER TECHNOLOGY CORPORATION (US) 2010-04-27 US disclosed
US-7410934-B2 Aqueous viscoelastic fluid SCHLUMBERGER TECHNOLOGY CORPORATION (US) 2008-08-12 US disclosed
US-20040102330-A1 Viscoelastic compositions SCHLUMBERGR TECHNOLOGY CORPORATION 2004-05-27 US disclosed
US-20040094301-A1 Aqueous viscoelastic fluid SCHLUMBERGER TECHNOLOGY CORPORATION 2004-05-20 US disclosed
EP-1360395-A1 VISCOELASTIC COMPOSITIONS Sofitech N.V. (BE) 2003-11-12 EP disclosed
WO-2002064945-A1 VISCOELASTIC COMPOSITIONS SOFITECH N.V. (BE) 2002-08-22 WO disclosed
WO-2002064947-A1 AQUEOUS VISCOELASTIC FLUID SOFITECH N.V. (BE) 2002-08-22 WO disclosed