SCHEMBL328281

SCHEMBL328281

CNC(=O)c1ccc(Nc2nc(SC)[nH]c(=O)c2C(=O)NN)cc1C

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
XDH P47989 9/20 0.38
GFER P55789 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
SLC22A12 Q96S37 1/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
TYK2 P29597 1/20 0.35
ALDH1A1 P00352 2/20 0.34
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
TP53 P04637 2/20 0.34
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34
PTK2 Q05397 1/20 0.33
THRB P10828 1/20 0.33
KLK7 P49862 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10126587 0.91 XDH (0.39) XDHGFERRXFP1SLC22A12JAK2
SCHEMBL10156468 0.83 XDH (0.39) XDHGFERRXFP1SLC22A12JAK2
SCHEMBL10126474 0.80 XDH (0.43) XDHGFERRXFP1SLC22A12ALDH1A1
SCHEMBL10156543 0.78 SYK (0.40) GFERKDM4EGAAPTK2KLK7
SCHEMBL10156479 0.78 XDH (0.41) XDHGFERRXFP1SLC22A12
SCHEMBL10156488 0.78 XDH (0.41) XDHGFERRXFP1SLC22A12
SCHEMBL10155939 0.78 XDH (0.39) XDHGFERRXFP1SLC22A12LMNA
SCHEMBL10126584 0.74 JAK2 (0.45) JAK2JAK1
SCHEMBL282772 0.73 GFER (0.43) XDHGFERRXFP1
SCHEMBL10126531 0.73 ALDH1A1 (0.42) XDHGFERRXFP1SLC22A12ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2428508-A1 DIAMINO HETEROCYCLIC CARBOXAMIDE COMPOUND Astellas Pharma Inc. (JP) 2012-03-14 EP disclosed