SCHEMBL3286364

SCHEMBL3286364

CCc1cc(C(C)c2cc(CC)c(O)c(CC)c2)cc(CC)c1O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.46
GABRB2 P47870 2/20 0.46
ALOX15 P16050 1/20 0.43
ALOX12 P18054 1/20 0.43
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
ESR1 P03372 2/20 0.37
ESR2 Q92731 2/20 0.37
PDCD1 Q15116 1/20 0.37
CD274 Q9NZQ7 1/20 0.37
FFAR1 O14842 2/20 0.35
DHFR P00374 1/20 0.35
BCL2L1 Q07817 1/20 0.33
CYP2D6 P10635 1/20 0.33
HDAC4 P56524 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
RNASEH1 O60930 1/20 0.32
SIRT1 Q96EB6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10687761 0.87 ALOX15 (0.38) GABRA1GABRB2ALOX15ALOX12CYP1A2
SCHEMBL31337454 0.86 GABRA1 (0.46) GABRA1GABRB2ALOX15ALOX12CYP1A2
SCHEMBL14461952 0.83 GABRA1 (0.48) GABRA1GABRB2ALOX15ALOX12CYP1A2
SCHEMBL6393256 0.82 CYP1A2 (0.55) GABRA1GABRB2ALOX15ALOX12CYP1A2
SCHEMBL3285883 0.82 HMGCR (0.38) GABRA1GABRB2ALOX15ALOX12ESR1
SCHEMBL3289296 0.79 GABRA1 (0.44) GABRA1GABRB2ALOX15ALOX12CYP1A2
SCHEMBL14997928 0.79 PRKCE (0.36) GABRA1GABRB2ALOX15ALOX12
SCHEMBL8843703 0.79 GABRA1 (0.40) GABRA1GABRB2ALOX15ALOX12CYP1A2
SCHEMBL2154505 0.76 HTT (0.52) ALOX15ALOX12
SCHEMBL920814 0.76 ESR1 (0.50) GABRA1GABRB2ALOX15ALOX12CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7718337-B2 Electrophotographic photoreceptor MITSUBISHI CHEMICAL CORPORATION (JP) 2010-05-18 US disclosed
US-20090081570-A1 ELECTROPHOTOGRAPHIC PHOTORECEPTOR MITSUBISHI CHEMICAL CORPORATION (JP) 2009-03-26 US disclosed
US-7473507-B2 Electrophotographic photoreceptor with polyester resin in photosensitive layer MITSUBISHI CHEMICAL CORPORATION (JP) 2009-01-06 US disclosed
US-20060073400-A1 Electrophotographic photoreceptor MITSUBISHI CHEMICAL CORPORATION (JP) 2006-04-06 US disclosed
US-6114487-A COATING AGENT, MOLDING MATERIAL, IMPROVED MOLD RELEASE DOW CORNING TORAY SILICONE CO., LTD. (JP) 2000-09-05 US disclosed
US-4789730-A Preparation of polycarbonate having reduced cyclic carbonate oligomer content THE DOW CHEMICAL COMPANY (US) 1988-12-06 US disclosed
US-4558118-A Two phase interfacial polycondensation polycarbonate process GENERAL ELECTRIC COMPANY (US) 1985-12-10 US disclosed
US-4533722-A COPPER CONTAINING COCATALYST GENERAL ELECTRIC COMPANY (US) 1985-08-06 US disclosed
US-4515936-A IONIC SURFACTANT GENERAL ELECTRIC COMPANY (US) 1985-05-07 US disclosed
US-4507436-A WITH MODIFIED POLYSTYRENE GENERAL ELECTRIC COMPANY (US) 1985-03-26 US disclosed
US-4471105-A HIGH MOLECULAR WEIGHT POLYMERS FROM STERICALLY HINDERED BISPHENOLS; REUSE AND CIRCULATION OF CATALYST GENERAL ELECTRIC COMPANY (US) 1984-09-11 US disclosed
US-4436876-A CONDENSATION POLYMERIZATION GENERAL ELECTRIC COMPANY (US) 1984-03-13 US disclosed
US-4384108-A Two-phase interfacial polycarbonate process GENERAL ELECTRIC COMPANY (US) 1983-05-17 US disclosed
US-4377662-A Block copolymers of polyphenylene oxides and sterically-hindered aromatic polycarbonates GENERAL ELECTRIC COMPANY (US) 1983-03-22 US disclosed
US-4374959-A Block copolymers of polyphenylene oxides and non-sterically-hindered high molecular weight aromatic polycarbonates GENERAL ELECTRIC COMPANY (US) 1983-02-22 US disclosed
US-4374233-A MOLDING MATERIALS; ENGINEERING THERMOPLASTICS GENERAL ELECTRIC COMPANY (US) 1983-02-15 US disclosed
US-4368315-A AGITATED TWO-PHASE MIXTURE OF ORGANIC SOLVENT AND WATER CONTAINING STRONG BASE GENERAL ELECTRIC COMPANY (US) 1983-01-11 US disclosed
US-4360659-A Non-catalyzed interfacial polycondensation polycarbonate process GENERAL ELECTRIC COMPANY (US) 1982-11-23 US disclosed
US-4345051-A Block copolymers of polyphenylene oxides and polyformals of sterically-hindered dihydric phenols GENERAL ELECTRIC COMPANY (US) 1982-08-17 US disclosed