SCHEMBL3289992

SCHEMBL3289992

Cc1cc(OC(F)(F)F)cc(C(=O)Nc2cccc(OC3CCN(C(=O)Nc4ccc(C(=O)O)cc4)CC3)c2)c1-c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 5/20 0.46
FAAH O00519 2/20 0.46
NR1H4 Q96RI1 2/20 0.44
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
NTRK1 P04629 1/20 0.42
KCNH2 Q12809 1/20 0.42
NTRK3 Q16288 1/20 0.42
NTRK2 Q16620 1/20 0.42
PRKAA2 P54646 1/20 0.42
POLB P06746 1/20 0.41
CFD P00746 1/20 0.41
NAMPT P43490 1/20 0.41
SCN9A Q15858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5144228 0.95 EPHX2 (0.45) EPHX2CYP2C9CYP2C19NTRK1KCNH2
SCHEMBL5142098 0.94 KMT2A (0.45) EPHX2CYP2C9CYP2C19NTRK1KCNH2
SCHEMBL4074904 0.90 EPHX2 (0.49) EPHX2FAAHCYP2C9CYP2C19NTRK1
SCHEMBL3290058 0.89 CFD (0.42) EPHX2NR1H4CYP2C9NTRK1KCNH2
SCHEMBL5145627 0.88 EPHX2 (0.43) EPHX2CYP2C9PRKAA2CFD
SCHEMBL3289653 0.87 EPHX2 (0.42) EPHX2FAAHCYP2C9PRKAA2CFD
SCHEMBL5298159 0.86 MAPT (0.44) PRKAA2POLB
SCHEMBL3288509 0.86 NTRK1 (0.50) EPHX2CYP2C9CYP2C19NTRK1KCNH2
SCHEMBL3295798 0.85 SLC5A7 (0.44) EPHX2CYP2C9PRKAA2CFD
SCHEMBL5143816 0.85 PRKAA2 (0.41) PRKAA2CFDSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7723358-B2 Aroyl-O-piperidine derivatives for the treatment of diabetes-related problems MERCK PATENT GMBH (DE) 2010-05-25 US claimed