SCHEMBL3295271

SCHEMBL3295271

C=C(C)O[C@H](C(=O)O)c1c(C)cc2nc(C3CC3)ccc2c1-c1ccc(Cl)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.35
PSIP1 O75475 1/20 0.35
PSD A5PKW4 5/20 0.34
FABP4 P15090 1/20 0.34
FABP5 Q01469 1/20 0.34
TRPC3 Q13507 1/20 0.33
TRPC7 Q9HCX4 1/20 0.33
DHODH Q02127 3/20 0.32
KDM4E B2RXH2 2/20 0.32
PLA2G2A P14555 1/20 0.32
MAPT P10636 3/20 0.32
ALDH1A1 P00352 2/20 0.32
HPGD P15428 2/20 0.32
NPSR1 Q6W5P4 2/20 0.32
MAPK1 P28482 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ADORA3 P0DMS8 1/20 0.31
NPC1 O15118 1/20 0.31
LMNA P02545 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3301651 0.87 CYP3A4 (0.36) CYP3A4PSIP1FABP4DHODHKDM4E
SCHEMBL245283 0.86 PSIP1 (0.49) CYP3A4PSIP1PSDFABP4FABP5
SCHEMBL10284000 0.85 KMT2A (0.35) CYP3A4PSIP1FABP4DHODHKDM4E
SCHEMBL27910448 0.83 DHODH (0.36) PSIP1PSDTRPC3TRPC7DHODH
SCHEMBL15182556 0.83 PSIP1 (0.41) CYP3A4PSIP1PSDFABP4FABP5
SCHEMBL10283998 0.83 EGLN1 (0.35) CYP3A4PSIP1DHODHKDM4EPLA2G2A
SCHEMBL15182618 0.83 CYP3A4 (0.40) CYP3A4PSIP1PSDFABP4FABP5
SCHEMBL10283992 0.82 KDM4E (0.39) CYP3A4PSIP1FABP4FABP5KDM4E
SCHEMBL3296191 0.82 GAA (0.35) CYP3A4PSIP1DHODHKDM4EPLA2G2A
SCHEMBL3312316 0.81 DHODH (0.33) CYP3A4PSIP1DHODHKDM4EPLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012003498-A1 2 -QUINOLINYL- ACETIC ACID DERIVATIVES AS HIV ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2012-01-05 WO disclosed