SCHEMBL3301651

SCHEMBL3301651

C=C(C)O[C@H](C(=O)O)c1c(C)cc2nc(C)ccc2c1-c1ccc(Cl)cc1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.36
PSIP1 O75475 1/20 0.36
DHODH Q02127 8/20 0.35
PLA2G2A P14555 1/20 0.35
POLB P06746 1/20 0.34
GRM2 Q14416 1/20 0.34
KDM4E B2RXH2 1/20 0.33
FABP3 P05413 1/20 0.33
FABP4 P15090 1/20 0.33
KMT2A Q03164 1/20 0.32
ADORA3 P0DMS8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10284000 0.90 KMT2A (0.35) CYP3A4PSIP1DHODHPLA2G2AGRM2
SCHEMBL10283998 0.88 EGLN1 (0.35) CYP3A4PSIP1DHODHPLA2G2APOLB
SCHEMBL3295271 0.87 CYP3A4 (0.35) CYP3A4PSIP1DHODHPLA2G2AKDM4E
SCHEMBL3296191 0.87 GAA (0.35) CYP3A4PSIP1DHODHPLA2G2AGRM2
SCHEMBL10284001 0.86 PLA2G2A (0.35) CYP3A4PSIP1DHODHPLA2G2AGRM2
SCHEMBL3296258 0.86 CYP3A4 (0.33) CYP3A4PSIP1DHODHPLA2G2AGRM2
SCHEMBL10283992 0.85 KDM4E (0.39) CYP3A4PSIP1POLBKDM4EFABP3
SCHEMBL244914 0.84 PSIP1 (0.51) CYP3A4PSIP1DHODHPOLBGRM2
SCHEMBL244717 0.84 PSIP1 (0.51) CYP3A4PSIP1DHODHPOLBGRM2
SCHEMBL3312316 0.84 DHODH (0.33) CYP3A4PSIP1DHODHPLA2G2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012003498-A1 2 -QUINOLINYL- ACETIC ACID DERIVATIVES AS HIV ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2012-01-05 WO disclosed