SCHEMBL3296191

SCHEMBL3296191

C=C(C)O[C@H](C(=O)O)c1c(C)cc2nc(C(=O)NC)ccc2c1-c1ccc(Cl)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.35
RAB9A P51151 1/20 0.35
SCN10A Q9Y5Y9 2/20 0.35
GRM2 Q14416 1/20 0.35
SCN1A P35498 1/20 0.35
KCNH2 Q12809 1/20 0.35
SCN5A Q14524 1/20 0.35
SCN9A Q15858 1/20 0.35
SCN2A Q99250 1/20 0.35
SCN3A Q9NY46 1/20 0.35
MALT1 Q9UDY8 5/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
PLA2G2A P14555 1/20 0.34
CYP3A4 P08684 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
PSIP1 O75475 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3301651 0.87 CYP3A4 (0.36) GRM2KMT2APLA2G2ACYP3A4PSIP1
SCHEMBL15186229 0.86 PSIP1 (0.47) GAARAB9ASCN10AGRM2SCN1A
SCHEMBL10284000 0.85 KMT2A (0.35) RAB9AGRM2MEN1KMT2APLA2G2A
SCHEMBL27928083 0.83 CNR1 (0.39) GAARAB9ASCN10AGRM2SCN1A
SCHEMBL10284001 0.83 PLA2G2A (0.35) GRM2SCN9AKMT2APLA2G2ACYP3A4
SCHEMBL10283998 0.83 EGLN1 (0.35) KMT2ANFKB1PLA2G2ACYP3A4SMN1; SMN2
SCHEMBL3295271 0.82 CYP3A4 (0.35) RAB9AMEN1KMT2APLA2G2ACYP3A4
SCHEMBL3296258 0.81 CYP3A4 (0.33) GRM2PLA2G2ACYP3A4PSIP1KDM4E
SCHEMBL10283992 0.80 KDM4E (0.39) GAACYP3A4PSIP1KDM4E
SCHEMBL3312316 0.80 DHODH (0.33) PLA2G2ACYP3A4PSIP1KDM4EDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012003498-A1 2 -QUINOLINYL- ACETIC ACID DERIVATIVES AS HIV ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2012-01-05 WO disclosed