SCHEMBL3309036

SCHEMBL3309036

COC(=O)c1cc2c(s1)CN(C)C(C)C2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.49
RAB9A P51151 5/20 0.49
KDM4E B2RXH2 5/20 0.49
HPGD P15428 5/20 0.49
MAPK1 P28482 3/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
HDAC6 Q9UBN7 2/20 0.42
ALDH1A1 P00352 6/20 0.42
L3MBTL1 Q9Y468 4/20 0.40
GLA P06280 2/20 0.38
GAA P10253 2/20 0.38
ATM Q13315 2/20 0.38
MAPT P10636 2/20 0.38
PKM P14618 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
TSHR P16473 2/20 0.37
HSD17B10 Q99714 2/20 0.37
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3314687 0.87 ALDH1A1 (0.45) NPC1RAB9AKDM4EHPGDHDAC6
SCHEMBL4436567 0.78 ALDH1A1 (0.33) NPC1RAB9AKDM4EHPGDMAPK1
SCHEMBL3310435 0.78 HPGD (0.55) NPC1RAB9AKDM4EHPGDMAPK1
SCHEMBL1174522 0.74 HDAC6 (0.53) NPC1RAB9AKDM4EHPGDMAPK1
SCHEMBL1397675 0.71 ALDH1A1 (0.53) NPC1RAB9AKDM4EHPGDMAPK1
SCHEMBL1173935 0.71 HDAC6 (0.60) NPC1RAB9AKDM4EHPGDMAPK1
SCHEMBL12922699 0.71 HDAC6 (0.53) NPC1RAB9AKDM4EHPGDMAPK1
Hydrochloric Acid SCHEMBL27148508 0.71 KDM4E (0.48) NPC1RAB9AKDM4EHPGDMAPK1
SCHEMBL3309479 0.71 KDM4E (0.54) NPC1RAB9AKDM4EHPGDMAPK1
SCHEMBL31670239 0.69 HDAC6 (0.61) NPC1RAB9AKDM4EHPGDMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8309542-B2 Substituted pyrrolidine amides, the production thereof, and the use thereof as medications BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-11-13 US disclosed
US-20100099664-A1 SUBSTITUTED PYRROLIDINE AMIDES, THE PRODUCTION THEREOF, AND THE USE THEREOF AS MEDICATIONS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100099664-A1 SUBSTITUTED PYRROLIDINE AMIDES, THE PRODUCTION THEREOF, AND THE USE THEREOF AS MEDICATIONS DDC, GLS, UROD NPC1 3523/4885RAB9A 2468/4885KDM4E 2370/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.