SCHEMBL332859

SCHEMBL332859

CCOC(=O)c1c(I)c(NC(C)=O)c(I)c(NC(C)=O)c1I

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.54
ALDH1A1 P00352 4/20 0.49
TSHR P16473 4/20 0.49
KDM4E B2RXH2 3/20 0.43
TP53 P04637 2/20 0.43
KMT2A Q03164 1/20 0.43
HPGD P15428 2/20 0.42
ALOX15 P16050 1/20 0.42
MAPT P10636 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
ALOX12 P18054 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
GAA P10253 1/20 0.41
PRKCZ Q05513 1/20 0.40
GLA P06280 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8814469 0.97 LMNA (0.50) LMNAALDH1A1TSHRKDM4ETP53
SCHEMBL28489419 0.91 LMNA (0.55) LMNAALDH1A1TSHRKDM4ETP53
SCHEMBL30018340 0.91 LMNA (0.55) LMNAALDH1A1TSHRKDM4ETP53
Ethyl Cartrizoate SCHEMBL2110540 0.89 LMNA (0.47) LMNAALDH1A1TSHRKDM4ETP53
Mannitol SCHEMBL8510041 0.87 SMN1; SMN2 (0.60) LMNAALDH1A1TSHRKDM4ETP53
Benzoic Acid SCHEMBL9410598 0.86 KDM4E (0.49) LMNAALDH1A1TSHRKDM4ETP53
SCHEMBL8752047 0.86 LMNA (0.44) LMNAALDH1A1TSHRKDM4ETP53
SCHEMBL9016334 0.85 LMNA (0.53) LMNAALDH1A1TSHRKDM4ETP53
SCHEMBL8230945 0.85 LMNA (0.53) LMNAALDH1A1TSHRKDM4ETP53
SCHEMBL371082 0.85 LMNA (0.46) LMNAALDH1A1TSHRKDM4ETP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 320 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2275094-A2 Reduction of intravenously administered nanoparticulate-formulation-induced adverse physiological reactions Elan Pharma International Limited (IE) 2011-01-19 EP claimed
US-20090081297-A1 Use of surface tension reducing agents in aerosol formulations MAP PHARMACEUTICALS, INC. 2009-03-26 US claimed
US-20050265923-A1 Embolus therapy using insoluble microparticles or vesicles containing contrast agents TONER JOHN L 2005-12-01 US claimed
US-20050258288-A1 High pressure media milling system and process of forming particles E. I. DU PONT DE NEMOURS AND COMPANY 2005-11-24 US claimed
WO-2005053851-A1 HIGH PRESSURE MEDIA MILLING SYSTEM AND PROCESS OF MILLING PARTICLES E.I. DUPONT DE NEMOURS AND COMPANY (US) 2005-06-16 WO claimed
EP-0810855-B1 POLYALKYLENE BLOCK COPOLYMERS AS SURFACE MODIFIERS FOR NANOPARTICLES ELAN PHARMA INT LTD (IE) 2003-06-11 EP claimed
EP-0804161-B1 CONTINUOUS METHOD OF GRINDING PHARMACEUTICAL SUBSTANCES ELAN PHARMA INT LTD (IE) 2001-11-07 EP claimed
EP-0804162-B1 BUTYLENE OXIDE-ETHYLENE OXIDE BLOCK COPOLYMER SURFACTANTS AS STABILIZER COATINGS FOR NANOCRYSTAL FORMULATION ELAN PHARMA INT LTD (IE) 2001-09-05 EP claimed
EP-0499299-B1 Surface modified drug nanoparticles NANOSYSTEMS LLC (US) 2000-08-16 EP claimed
EP-0600528-B1 Method of grinding pharmaceutical substances ELAN PHARMA INTERNATIONAL LIMI (IE) 2000-06-07 EP claimed
EP-0602700-A2 Novel formulations for nanoparticulate X-ray blood pool contrast agents using high molecular weight surfactants NanoSystems L.L.C. (US) 1994-06-22 EP claimed
EP-0601619-A2 Use of non-ionic cloud point modifiers to minimize nanoparticle aggregation during sterilization NanoSystems L.L.C. (US) 1994-06-15 EP claimed
EP-0600528-A1 Method of grinding pharmaceutical substances NanoSystems L.L.C. (US) 1994-06-08 EP claimed
EP-0600532-A2 Use of ionic cloud point modifiers to prevent particle aggregation during sterilization NanoSystems L.L.C. (US) 1994-06-08 EP claimed
US-5318768-A For gastrointestinal tract; film membrane, cation potentiator, particle surface modifier STERLING WINTHROP INC. (US) 1994-06-07 US claimed
US-5318767-A X-ray contrast compositions useful in medical imaging STERLING WINTHROP INC. (US) 1994-06-07 US claimed
US-5298262-A Nonionic surfactant particles STERLING WINTHROP INC. (US) 1994-03-29 US claimed
US-5145684-A SURFACE MODIFIED DRUG NANOPARTICLES STERLING DRUG INC. (US) 1992-09-08 US claimed
EP-0499299-A2 Surface modified drug nanoparticles NanoSystems L.L.C. (US) 1992-08-19 EP claimed
EP-0498482-A2 X-ray contrast compositions useful in medical imaging NanoSystems L.L.C. (US) 1992-08-12 EP claimed