Chlorpheniramine

Chlorpheniramine

SCHEMBL33358

CN(C)CC[C@H](c1ccc(Cl)cc1)c1ccccn1.O=C(O)C=CC(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

HRH1

The experimentally established mechanism targets of Chlorpheniramine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 known ✓ P35367 5/20 0.81
LMNA P02545 4/20 1.00
PMP22 Q01453 2/20 1.00
BLM P54132 1/20 1.00
NPSR1 Q6W5P4 1/20 1.00
TSHR P16473 2/20 0.84
ALDH1A1 P00352 1/20 0.84
CYP3A4 P08684 1/20 0.84
CYP2C19 P33261 1/20 0.84
KDM4E B2RXH2 1/20 0.84
RAB9A P51151 1/20 0.84
CHRM2 P08172 6/20 0.81
SLC6A2 P23975 6/20 0.81
SLC6A4 P31645 6/20 0.81
SLC6A3 Q01959 5/20 0.81
KCNH2 Q12809 5/20 0.81
HRH3 Q9Y5N1 5/20 0.81
CHRM1 P11229 4/20 0.81
ADRA2B P18089 4/20 0.81
HTR2A P28223 3/20 0.81

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Chlorpheniramine SCHEMBL14973510 1.00 LMNA (1.00) LMNAPMP22BLMNPSR1TSHR
Chlorpheniramine SCHEMBL30487016 1.00 LMNA (1.00) LMNAPMP22BLMNPSR1TSHR
Dexchlorpheniramine SCHEMBL119500 1.00 LMNA (1.00) LMNAPMP22BLMNPSR1TSHR
Chlorpheniramine SCHEMBL27719385 1.00 LMNA (1.00) LMNAPMP22BLMNPSR1TSHR
Chlorpheniramine SCHEMBL4359260 1.00 LMNA (1.00) LMNAPMP22BLMNPSR1TSHR
Chlorpheniramine SCHEMBL33357 1.00 LMNA (1.00) LMNAPMP22BLMNPSR1TSHR
Chlorpheniramine SCHEMBL4284232 0.99 LMNA (0.98) LMNAPMP22BLMNPSR1TSHR
Chlorpheniramine SCHEMBL4284230 0.99 LMNA (0.98) LMNAPMP22BLMNPSR1TSHR
Chlorpheniramine SCHEMBL28130816 0.99 LMNA (0.98) LMNAPMP22BLMNPSR1TSHR
Chlorpheniramine SCHEMBL10002622 0.99 LMNA (0.98) LMNAPMP22BLMNPSR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 10897 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122076970-A Platinum iridium bimetallic nano-enzyme, preparation method and application thereof in immunochromatography detection 2026-05-26 CN claimed
US-12629422-B2 Agave syrup formulation or suspension for active pharmaceutical agents GENEXA INC. (US) 2026-05-19 US claimed
EP-4734952-A1 ORAL TABLET WITH IMPROVED UNIFORMITY OF CONTENT OF ACTIVES Fertin Pharma A/S (DK) 2026-05-06 EP claimed
US-20260090584-A1 SYSTEMS AND METHODS FOR ESTIMATING AEROSOLIZATION EMISSION SCIENTIFIC HORIZONS CONSULTING LLC (US) 2026-04-02 US claimed
US-20260041675-A1 NASAL COMPOSITION SATO PHARMACEUTICAL CO., LTD. (JP) 2026-02-12 US claimed
US-20250367139-A1 COMPOUND HYDROCORTISONE AND NEOMYCIN SULFATE GRANULE AND PREPARATION METHOD THEREOF HEBEI CHANGTIAN PHARMACEUTICAL CO LTD (CN) 2025-12-04 US claimed
EP-4654949-A1 USE OF VITAMIN E TPGS AS A TASTE MASKING AGENT FOR BITTER DRUGS Hyloris Developments SA (BE) 2025-12-03 EP claimed
US-20250332120-A1 COMPOSITION FOR EXTERNAL PREPARATION KAO CORPORATION (JP) 2025-10-30 US claimed
US-20250325483-A1 FLOWPACK WITH COMPOSITION FOR IMPROVED TASTE MASKING OF ACTIVES FERTIN PHARMA AS (DK) 2025-10-23 US claimed
US-20250312272-A1 PHARMACEUTICAL FORMULATIONS FOR ORAL ADMINISTRATION AND METHODS OF MAKING AND USING THE SAME Brunswick Pharma LLC 2025-10-09 US claimed
EP-0189861-A2 Percutaneous absorption accelerator for ionic water-soluble medicine SHOWA DENKO KABUSHIKI KAISHA (JP) 1986-08-06 EP claimed
US-4576645-A Whipped gel composition BLOCK DRUG CO., INC. (US) 1986-03-18 US claimed
EP-0132472-A1 Medicated products containing a magnesium trisilicate adsorbent with a medicament drug adsorbed thereon WARNER-LAMBERT COMPANY (US) 1985-02-13 EP claimed
US-4472372-A Polymeric diffusion matrix containing chlorpheniramine maleate KEY PHARMACEUTICALS, INC. (US) 1984-09-18 US claimed
US-4455146-A THERMOPLASTIC ELASTOMERS, OILS OR FATTY ACID, TACKFIER, AND A MEDICINE HISAMITSU PHARMACEUTICAL CO., LTD. (JP) 1984-06-19 US claimed
EP-0079545-A1 Benzimidazole derivatives, process for the preparation thereof and pharmaceutical composition containing the same KANEBO, LTD. (JP) 1983-05-25 EP claimed
WO-1982000099-A1 POLYMERIC DIFFUSION MATRIX FOR ADMINISTRATION OF DRUGS KEY PHARMA (US) 1982-01-21 WO claimed
US-4278679-A ANTIHISTAMINE, PREVENTION OF ANTICHOLINERGIC EFFECT CHROMALLOY AMERICAN CORPORATION (US) 1981-07-14 US claimed
US-4269835-A Nasal composition for relieving nasal distress WHITTLE BARRY J 1981-05-26 US claimed
US-4256763-A ANTIINFLAMMATORY AGENTS, VIRICIDES, PHENOLPHTHALEIN MCHUGH JOHN E 1981-03-17 US claimed