SCHEMBL3341252

SCHEMBL3341252

O=C(O)c1c[nH]c2cc(N3CCNCC3)c(F)cc2c1=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.58
HPGD P15428 6/20 0.58
HSD17B10 Q99714 6/20 0.58
ALDH1A1 P00352 6/20 0.58
LMNA P02545 5/20 0.58
TOP2A P11388 4/20 0.58
TOP2B Q02880 3/20 0.58
CYP2C9 P11712 2/20 0.58
CYP1A2 P05177 2/20 0.58
BRD4 O60885 1/20 0.58
TSHR P16473 1/20 0.58
HTT P42858 1/20 0.58
CYP2J2 P51589 1/20 0.58
NPSR1 Q6W5P4 1/20 0.58
ATP6V1B2 P21281 1/20 0.46
TBXA2R P21731 1/20 0.46
EDNRA P25101 1/20 0.46
TARBP2 Q15633 1/20 0.46
MEN1 O00255 3/20 0.45
KMT2A Q03164 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cyclopropane SCHEMBL3447310 0.98 ALDH1A1 (0.56) KDM4EHPGDHSD17B10ALDH1A1LMNA
SCHEMBL3401906 0.90 KDM4E (0.52) KDM4EHPGDHSD17B10ALDH1A1LMNA
SCHEMBL17475410 0.89 KDM4E (0.51) KDM4EHPGDHSD17B10ALDH1A1LMNA
SCHEMBL10743065 0.88 KDM4E (0.50) KDM4EHPGDHSD17B10ALDH1A1LMNA
SCHEMBL9379704 0.87 ALDH1A1 (0.58) KDM4EHPGDHSD17B10ALDH1A1LMNA
SCHEMBL5307312 0.87 KDM4E (0.49) KDM4EHPGDHSD17B10ALDH1A1LMNA
SCHEMBL9626251 0.85 KDM4E (0.47) KDM4EHPGDHSD17B10ALDH1A1LMNA
SCHEMBL7557789 0.84 ALDH1A1 (0.50) KDM4EHPGDHSD17B10ALDH1A1LMNA
SCHEMBL6714523 0.82 HPGD (0.45) KDM4EHPGDHSD17B10ALDH1A1LMNA
SCHEMBL21111089 0.82 HSD17B10 (0.51) KDM4EHPGDHSD17B10ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1990000551-A1 PROCESS FOR THE PREPARATION OF QUINOLINE ANTIBACTERIAL COMPOUNDS ABBOTT LABORATORIES (US) 1990-01-25 WO claimed
EP-0350950-A1 Process for the preparation of quinoline antibacterial compounds ABBOTT LABORATORIES (US) 1990-01-17 EP claimed
US-20100094230-A1 POLYMER MOLDING COMPOUNDS CONTAINING PARTIALLY NEUTRALIZED AGENTS BAYER INNOVATION GMBH (DE) 2010-04-15 US disclosed