SCHEMBL334470

SCHEMBL334470

Ic1cc(-c2cccnn2)no1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.33
GOT1 P17174 1/20 0.31
DHODH Q02127 1/20 0.31
HTR2C P28335 1/20 0.31
CYP1A2 P05177 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4046101 0.77 KDM4E (0.54) GRM5CYP1A2SMN1; SMN2
SCHEMBL29442588 0.76 GOT1 (0.46) GRM5GOT1DHODHHTR2CCYP1A2
SCHEMBL1456807 0.76 GOT1 (0.46) GRM5GOT1DHODHHTR2CCYP1A2
SCHEMBL30792004 0.76 GOT1 (0.46) GRM5GOT1DHODHHTR2CCYP1A2
SCHEMBL10282499 0.75 CYP2E1 (0.39) HTR2CSMN1; SMN2
SCHEMBL11849360 0.75 RAB9A (0.42) SMN1; SMN2
SCHEMBL27790048 0.75 SMN1; SMN2 (0.39) GRM5DHODHCYP1A2SMN1; SMN2
SCHEMBL27790050 0.75 DHODH (0.34) GRM5DHODH
SCHEMBL10243416 0.75 MEN1 (0.56) SMN1; SMN2
SCHEMBL12571308 0.74 HCAR2 (0.43) DHODHCYP1A2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8097708-B2 10a-Azalide compound TAISHO PHARMACEUTICAL CO., LTD. (JP) 2012-01-17 US disclosed
US-20090281292-A1 10a-Azalide Compound MEIJI SEIKA PHARMA CO., LTD. (JP) 2009-11-12 US disclosed
EP-1985620-A1 10a-AZALIDE COMPOUND TAISHO PHARMACEUTICAL CO., LTD (JP) 2008-10-29 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090281292-A1 10a-Azalide Compound IL17A, AZI2, HDAC9 GRM5 4381/4885GOT1 4102/4885DHODH 1930/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.