SCHEMBL3345117

SCHEMBL3345117

COC(=O)COc1ccc(F)c2c1c(C)c(Cc1ccc(-n3cccn3)cc1)c(=O)n2C

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 1/20 0.50
CHRM1 P11229 7/20 0.38
KDM4E B2RXH2 1/20 0.38
JAK2 O60674 1/20 0.38
RORC P51449 9/20 0.37
KLKB1 P03952 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3344793 0.93 PTGDR2 (0.58) PTGDR2CHRM1RORCKLKB1CYP3A4
SCHEMBL3351455 0.90 PTGDR2 (0.43) PTGDR2CHRM1RORCKLKB1CYP3A4
SCHEMBL3344721 0.84 P2RX3 (0.42) PTGDR2KDM4EJAK2
SCHEMBL2571339 0.84 PTGDR2 (0.50) PTGDR2CHRM1KDM4EJAK2RORC
SCHEMBL3345546 0.82 PTGDR2 (0.50) PTGDR2CHRM1RORCKLKB1CYP3A4
SCHEMBL2575061 0.82 PTGDR2 (0.56) PTGDR2RORC
SCHEMBL3346044 0.81 TSHR (0.37) PTGDR2KDM4EJAK2
SCHEMBL2570536 0.81 PTGDR2 (0.56) PTGDR2CHRM1KDM4EJAK2RORC
SCHEMBL2570380 0.80 PTGDR2 (0.55) PTGDR2CHRM1RORC
SCHEMBL2568426 0.79 PTGDR2 (0.62) PTGDR2CHRM1RORCKLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010040989-A1 QUINOLIN-2-ONE COMPOUNDS ARGENTA ORAL THERAPEUTICS LIMITED (GB) 2010-04-15 WO disclosed