SCHEMBL3345496

SCHEMBL3345496

Cc1ccc(-c2sc(N(C)C)nc2C(=O)O)cc1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.45
HCRTR1 O43613 4/20 0.38
HCRTR2 O43614 4/20 0.38
AKR1C3 P42330 2/20 0.37
AKR1C2 P52895 2/20 0.37
GRIN2B Q13224 1/20 0.36
AKR1B10 O60218 1/20 0.36
AKR1C4 P17516 1/20 0.36
AKR1C1 Q04828 1/20 0.36
XDH P47989 1/20 0.35
SLC22A12 Q96S37 1/20 0.35
NISCH Q9Y2I1 1/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
PIK3CG P48736 1/20 0.34
ERN1 O75460 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL984634 0.88 HCRTR1 (0.45) HCRTR1HCRTR2ALDH1A1HPGD
SCHEMBL984476 0.84 KMO (0.49) KMOHCRTR1HCRTR2AKR1C3AKR1C2
SCHEMBL980677 0.83 PIN1 (0.50) KMO
SCHEMBL984151 0.82 MAPK14 (0.41) HCRTR1HCRTR2ALDH1A1HPGDHSD17B10
SCHEMBL27834590 0.81 KDM4E (0.44) HCRTR1HCRTR2ALDH1A1HPGDHSD17B10
SCHEMBL14850865 0.81 NISCH (0.40) KMOGRIN2BNISCHPIK3CDPIK3CA
SCHEMBL1340321 0.79 PIN1 (0.49) KMOHCRTR1HCRTR2ALDH1A1HPGD
SCHEMBL980993 0.78 ALDH1A1 (0.47) HCRTR1HCRTR2ALDH1A1HPGDHSD17B10
SCHEMBL984955 0.78 HCRTR1 (0.49) KMOHCRTR1HCRTR2AKR1C3AKR1C2
SCHEMBL984890 0.77 HCRTR1 (0.38) HCRTR1HCRTR2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102164896-A Phenethylamide derivatives and their heterocyclic analogues ACTELION PHARMACEUTICALS LTD 2011-08-24 CN claimed
WO-2010044054-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES ACTELION PHARMACEUTICALS LTD (CH) 2010-04-22 WO claimed
CN-102164896-A Phenethylamide derivatives and their heterocyclic analogues ACTELION PHARMACEUTICALS LTD 2011-08-24 CN disclosed
WO-2010044054-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES ACTELION PHARMACEUTICALS LTD (CH) 2010-04-22 WO disclosed