SCHEMBL3345948

SCHEMBL3345948

Cc1ccc(-c2nccnc2C(=O)N2CCOC2C(N)=O)cc1C

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 11/20 0.38
HCRTR1 O43613 10/20 0.38
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
MAPK1 P28482 1/20 0.38
PDE10A Q9Y233 1/20 0.34
EGFR P00533 1/20 0.32
GRIN2B Q13224 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3350896 0.86 HCRTR1 (0.51) HCRTR2HCRTR1PDE10AGRIN2B
SCHEMBL3345952 0.84 HCRTR1 (0.38) HCRTR2HCRTR1ALDH1A1MEN1KMT2A
SCHEMBL3343763 0.79 HCRTR1 (0.49) HCRTR2HCRTR1
SCHEMBL2635182 0.79 HCRTR1 (0.38) HCRTR2HCRTR1ALDH1A1MEN1KMT2A
SCHEMBL3350764 0.76 HCRTR1 (0.50) HCRTR2HCRTR1
SCHEMBL3350490 0.76 HCRTR1 (0.43) HCRTR2HCRTR1ALDH1A1MEN1KMT2A
SCHEMBL2056953 0.74 KCNA5 (0.39) HCRTR2HCRTR1ALDH1A1MEN1KMT2A
SCHEMBL984761 0.72 MCL1 (0.46) ALDH1A1MEN1KMT2AMAPK1
SCHEMBL3350904 0.71 HCRTR1 (0.51) HCRTR2HCRTR1PDE10AGRIN2B
SCHEMBL2635825 0.70 PDE10A (0.40) HCRTR2HCRTR1PDE10AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038200-A1 OXAZOLIDINE COMPOUNDS AS OREXIN RECEPTOR ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2010-04-08 WO claimed
WO-2010038200-A1 OXAZOLIDINE COMPOUNDS AS OREXIN RECEPTOR ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2010-04-08 WO disclosed