SCHEMBL3350896

SCHEMBL3350896

Cc1cccc(-c2nccnc2C(=O)N2CCOC2C(N)=O)c1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 8/20 0.51
HCRTR2 O43614 8/20 0.51
PDE10A Q9Y233 4/20 0.38
GRIN2B Q13224 1/20 0.36
RIPK2 O43353 1/20 0.36
KMO O15229 1/20 0.35
TLR8 Q9NR97 1/20 0.35
KDM5A P29375 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
NR3C2 P08235 1/20 0.35
GRM5 P41594 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3345948 0.86 HCRTR2 (0.38) HCRTR1HCRTR2PDE10AGRIN2B
SCHEMBL3350904 0.84 HCRTR1 (0.51) HCRTR1HCRTR2PDE10AGRIN2B
SCHEMBL3344465 0.80 HCRTR1 (0.51) HCRTR1HCRTR2
SCHEMBL2635740 0.79 HCRTR1 (0.51) HCRTR1HCRTR2PDE10ARIPK2TLR8
SCHEMBL2056990 0.74 HCRTR1 (0.51) HCRTR1HCRTR2PDE10AGRIN2B
SCHEMBL2057011 0.73 KMO (0.52) HCRTR1HCRTR2KMOKDM5AKDM4C
SCHEMBL3344316 0.72 HCRTR1 (0.46) HCRTR1HCRTR2
SCHEMBL3345952 0.71 HCRTR1 (0.38) HCRTR1HCRTR2GRIN2B
SCHEMBL3348002 0.68 HCRTR1 (0.44) HCRTR1HCRTR2
SCHEMBL3344362 0.67 HCRTR1 (0.53) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010038200-A1 OXAZOLIDINE COMPOUNDS AS OREXIN RECEPTOR ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2010-04-08 WO claimed
WO-2010038200-A1 OXAZOLIDINE COMPOUNDS AS OREXIN RECEPTOR ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2010-04-08 WO disclosed