SCHEMBL3346294

SCHEMBL3346294

COc1ccc(CCC(C(N)=O)N(C)C)cc1OC

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 1/20 0.56
AOC3 Q16853 1/20 0.54
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2D6 P10635 1/20 0.53
KDM4E B2RXH2 2/20 0.51
ATM Q13315 1/20 0.51
BLM P54132 1/20 0.51
PMP22 Q01453 1/20 0.51
LDHA P00338 1/20 0.50
CYP19A1 P11511 1/20 0.49
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA9 Q16790 1/20 0.48
ALDH1A1 P00352 2/20 0.47
KMT2A Q03164 2/20 0.47
CDK8 P49336 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3348404 0.81 STAT3 (0.65) STAT3AOC3KDM4EATMLDHA
SCHEMBL3351884 0.79 STAT3 (0.59) STAT3AOC3CYP1A2CYP3A4CYP2D6
SCHEMBL5192260 0.78 STAT3 (0.57) STAT3AOC3KDM4EATMLDHA
SCHEMBL29378321 0.77 LDHA (0.60) STAT3AOC3KDM4EATMLDHA
SCHEMBL29965330 0.77 LDHA (0.60) STAT3AOC3KDM4EATMLDHA
SCHEMBL22445062 0.75 STAT3 (0.57) STAT3KDM4EATMLDHACYP19A1
SCHEMBL27673600 0.75 STAT3 (0.71) STAT3AOC3CYP1A2CYP3A4CYP2D6
SCHEMBL6093053 0.75 KMT2A (0.57) STAT3KDM4EATMLDHAALDH1A1
SCHEMBL3578334 0.75 STAT3 (0.87) STAT3AOC3CYP1A2CYP3A4CYP2D6
SCHEMBL10927650 0.75 STAT3 (0.47) STAT3AOC3CYP3A4KDM4EATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010044054-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES ACTELION PHARMACEUTICALS LTD (CH) 2010-04-22 WO claimed
WO-2010044054-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES ACTELION PHARMACEUTICALS LTD (CH) 2010-04-22 WO disclosed