SCHEMBL3346487

SCHEMBL3346487

CC(C)(C)c1ccc([C@@H]2CNC[C@H]2C(=O)NCCc2ccccc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MC4R P32245 5/20 0.59
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
ESRRG P62508 2/20 0.52
TAAR1 Q96RJ0 4/20 0.52
KCNH2 Q12809 4/20 0.52
POLB P06746 1/20 0.48
GAA P10253 1/20 0.48
KDM1A O60341 1/20 0.47
MAOA P21397 1/20 0.46
SSTR4 P31391 1/20 0.45
TLR2 O60603 1/20 0.44
TLR1 Q15399 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346236 0.89 MC4R (0.65) MC4RTAAR1KCNH2POLBGAA
SCHEMBL3346234 0.88 MC4R (0.71) MC4RTAAR1KCNH2POLBGAA
SCHEMBL3346376 0.85 MC4R (0.63) MC4RNPC1RAB9ATAAR1KCNH2
SCHEMBL3353035 0.81 MC4R (0.56) MC4RTAAR1KCNH2POLBGAA
SCHEMBL3348167 0.81 MC4R (0.60) MC4RTAAR1KCNH2POLBGAA
SCHEMBL22178742 0.80 MC4R (0.88) MC4RTAAR1POLBGAA
SCHEMBL3353142 0.79 MC4R (0.62) MC4RTAAR1POLBGAATLR2
Hydrochloric Acid SCHEMBL22160650 0.79 MC4R (0.86) MC4RTAAR1POLBGAA
SCHEMBL3410126 0.78 MC4R (0.57) MC4RNPC1RAB9ATAAR1KCNH2
SCHEMBL3348194 0.78 KCNH2 (0.63) MC4RTAAR1KCNH2POLBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed