SCHEMBL3353142

SCHEMBL3353142

O=C(NCCc1ccccc1)[C@@H]1CNC[C@H]1c1cc(Cl)cc(Cl)c1

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MC4R P32245 5/20 0.62
TAAR1 Q96RJ0 7/20 0.53
GLA P06280 1/20 0.52
ALDH1A1 P00352 3/20 0.50
CASP1 P29466 1/20 0.50
HSD17B10 Q99714 1/20 0.50
POLB P06746 1/20 0.50
GAA P10253 1/20 0.50
SCN9A Q15858 1/20 0.43
HPGD P15428 1/20 0.43
TLR2 O60603 1/20 0.43
TLR1 Q15399 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
MAPT P10636 1/20 0.43
NLRP3 Q96P20 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3353265 0.93 MC4R (0.53) MC4RTAAR1GLAALDH1A1
SCHEMBL3346679 0.91 MC4R (0.59) MC4RTAAR1GLAALDH1A1CASP1
SCHEMBL3346376 0.89 MC4R (0.63) MC4RTAAR1GLAALDH1A1CASP1
SCHEMBL3353136 0.88 TAAR1 (0.50) MC4RTAAR1GLAALDH1A1CASP1
SCHEMBL3346234 0.87 MC4R (0.71) MC4RTAAR1ALDH1A1POLBGAA
SCHEMBL3347960 0.85 CNR1 (0.52) MC4RTAAR1GLAALDH1A1POLB
SCHEMBL3349847 0.83 MC4R (0.58) MC4RTAAR1GLAALDH1A1CASP1
SCHEMBL3348167 0.82 MC4R (0.60) MC4RTAAR1ALDH1A1POLBGAA
SCHEMBL3346447 0.82 MC4R (0.63) MC4RTAAR1GLAALDH1A1CASP1
SCHEMBL3410126 0.82 MC4R (0.57) MC4RTAAR1POLBGAATLR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed