SCHEMBL3353119

SCHEMBL3353119

Cc1cccc([C@H](C)NC(=O)[C@@H]2CNC[C@H]2c2ccc(C(F)(F)F)cn2)n1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 5/20 0.47
PDE2A O00408 2/20 0.42
GPR139 Q6DWJ6 1/20 0.35
SSTR4 P31391 3/20 0.35
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34
SCN9A Q15858 1/20 0.34
ACACB O00763 1/20 0.34
ACKR3 P25106 2/20 0.34
FFAR1 O14842 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346552 0.89 KCNH2 (0.45) KCNH2PDE2AGPR139SCN9AACACB
SCHEMBL3346452 0.87 KCNH2 (0.48) KCNH2PDE2AGPR139SSTR4ACACB
SCHEMBL3346544 0.86 TRPM5 (0.38) KCNH2SSTR4ACKR3
SCHEMBL13365135 0.84 KCNH2 (0.57) KCNH2PDE2AGPR139SCN9AACACB
SCHEMBL3346217 0.84 KCNH2 (0.51) KCNH2PDE2AGPR139SSTR4ACACB
SCHEMBL3346572 0.82 KCNH2 (0.51) KCNH2PDE2AACACB
SCHEMBL3346727 0.82 KCNH2 (0.53) KCNH2SSTR4PSEN1PSEN2APH1B
SCHEMBL3346554 0.81 KCNH2 (0.48) KCNH2PDE2ASSTR4ACACB
SCHEMBL3346567 0.81 KCNH2 (0.59) KCNH2PDE2AACACB
SCHEMBL3346383 0.81 KCNH2 (0.50) KCNH2PDE2AACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed