SCHEMBL3345898

SCHEMBL3345898

C[C@H](NC(=O)[C@@H]1CNC[C@H]1c1ccc(C(F)(F)F)nc1)c1ccccc1F

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.54
HDAC4 P56524 1/20 0.40
TRPM8 Q7Z2W7 1/20 0.40
SSTR4 P31391 1/20 0.37
TRPV1 Q8NER1 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
P2RX7 Q99572 1/20 0.36
ROCK2 O75116 2/20 0.35
ROCK1 Q13464 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3348192 0.87 KCNH2 (0.57) KCNH2HDAC4TRPM8
SCHEMBL13365071 0.87 KCNH2 (0.43) KCNH2SSTR4ROCK2ROCK1
SCHEMBL13365134 0.85 KCNH2 (0.64) KCNH2TRPM8SSTR4
SCHEMBL3346204 0.85 KCNH2 (0.54) KCNH2HDAC4TRPM8SSTR4HRH3
SCHEMBL3415190 0.85 KCNH2 (0.59) KCNH2HDAC4HRH3P2RX7ROCK2
SCHEMBL3347928 0.83 KCNH2 (0.53) KCNH2HDAC4TRPM8ROCK2
SCHEMBL3346727 0.81 KCNH2 (0.53) KCNH2HDAC4TRPM8SSTR4HRH3
SCHEMBL3346554 0.81 KCNH2 (0.48) KCNH2HDAC4TRPM8SSTR4ROCK2
SCHEMBL3346410 0.81 KCNH2 (0.48) KCNH2SSTR4ROCK2
SCHEMBL3350867 0.81 KCNH2 (0.52) KCNH2TRPM8TRPV1P2RX7ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed