SCHEMBL3346563

SCHEMBL3346563

Cc1ccsc1C#Cc1ccn2nccc2n1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.45
OGA O60502 1/20 0.40
DYRK1A Q13627 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
TGFBR1 P36897 2/20 0.33
FFAR1 O14842 1/20 0.33
KDM4E B2RXH2 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
HTT P42858 1/20 0.32
RECQL P46063 1/20 0.32
SCN5A Q14524 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3347616 0.79 DYRK1A (0.40) CYP2A6OGADYRK1AALDH1A1HPGD
SCHEMBL3347593 0.78 OGA (0.42) OGADYRK1ATGFBR1SCN5A
SCHEMBL3347052 0.78 CYP2A6 (0.37) CYP2A6OGADYRK1AALDH1A1HPGD
SCHEMBL3347020 0.77 CYP2A6 (0.36) CYP2A6OGAALDH1A1HPGDTGFBR1
SCHEMBL3348818 0.76 GRM5 (0.47) OGADYRK1ATGFBR1FFAR1SCN5A
SCHEMBL3346192 0.76 GRM5 (0.47) OGADYRK1ATGFBR1SCN5A
SCHEMBL3346766 0.76 GRM5 (0.53) ALDH1A1HPGDTGFBR1KDM4ECYP1A2
SCHEMBL3346384 0.74 GRM5 (0.43) OGADYRK1AALDH1A1HPGDTGFBR1
SCHEMBL3346767 0.72 GRM5 (0.46) CYP2A6OGADYRK1ASCN5A
SCHEMBL3351201 0.72 OGA (0.37) OGADYRK1ATGFBR1SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO claimed
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed