SCHEMBL3348554

SCHEMBL3348554

Cc1ccc2nc(NC(=O)c3cc[c]cc3)sc2c1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 1/20 0.72
DYRK1A Q13627 1/20 0.65
NPC1 O15118 11/20 0.64
RAB9A P51151 11/20 0.64
ALDH1A1 P00352 6/20 0.64
SMN1; SMN2 Q16637 6/20 0.64
KDM4E B2RXH2 5/20 0.64
HPGD P15428 4/20 0.64
KLK7 P49862 1/20 0.64
TDP1 Q9NUW8 1/20 0.64
LRRK2 Q5S007 1/20 0.62
MEN1 O00255 6/20 0.61
KMT2A Q03164 6/20 0.61
MAPT P10636 3/20 0.61
NFKB1 P19838 2/20 0.61
NFKB2 Q00653 2/20 0.61
RELA Q04206 2/20 0.61
TP53 P04637 2/20 0.61
OPRK1 P41145 1/20 0.61
HTT P42858 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13329390 0.89 MAP3K5 (0.83) MAP3K5DYRK1ANPC1RAB9AALDH1A1
SCHEMBL5713530 0.87 MAP3K5 (0.75) MAP3K5DYRK1ANPC1RAB9AALDH1A1
SCHEMBL2483622 0.86 MAP3K5 (0.77) MAP3K5DYRK1ANPC1RAB9AALDH1A1
SCHEMBL3347489 0.85 MAP3K5 (0.63) MAP3K5DYRK1ANPC1RAB9AALDH1A1
SCHEMBL12199362 0.85 MAP3K5 (0.76) MAP3K5DYRK1ANPC1RAB9AALDH1A1
SCHEMBL12225800 0.85 MAP3K5 (0.76) MAP3K5DYRK1ANPC1RAB9AALDH1A1
SCHEMBL12199335 0.85 MAP3K5 (0.76) MAP3K5DYRK1ANPC1RAB9AALDH1A1
SCHEMBL2485047 0.84 SCD (0.82) DYRK1ANPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL3347250 0.84 RAB9A (0.67) MAP3K5DYRK1ANPC1RAB9AALDH1A1
SCHEMBL12199491 0.82 MAP3K5 (0.72) MAP3K5DYRK1ANPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010066357-A1 BENZOTHIAZOLE AMIDES FOR DETECTION OF AMYLOID BETA BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-06-17 WO disclosed