SCHEMBL3348936

SCHEMBL3348936

Cc1csc(-c2nc(N)c3cc(CC(C)c4ccccn4)sc3n2)n1

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 19/20 0.64
ADORA1 P30542 16/20 0.64
PDE10A Q9Y233 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3297128 0.83 ADORA2A (0.74) ADORA2AADORA1
SCHEMBL3348932 0.82 ADORA2A (0.64) ADORA2AADORA1PDE10A
SCHEMBL13389506 0.82 ADORA2A (0.64) ADORA2AADORA1PDE10A
SCHEMBL3344541 0.81 ADORA2A (0.63) ADORA2AADORA1
SCHEMBL3350946 0.81 ADORA2A (0.64) ADORA2AADORA1
Hydrochloric Acid SCHEMBL3298338 0.81 ADORA2A (0.63) ADORA2AADORA1PDE10A
SCHEMBL3344914 0.80 ADORA2A (0.64) ADORA2AADORA1
Hydrochloric Acid SCHEMBL3345119 0.80 ADORA2A (0.63) ADORA2AADORA1PDE10A
SCHEMBL3300401 0.78 ADORA2A (1.00) ADORA2AADORA1
SCHEMBL3346316 0.77 ADORA2A (0.82) ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010045015-A1 HETEROARYL SUBSTITUTED THIENO[2,3-D]PYRIMIDINE AND THEIR USE AS ADENOSINE A2A RECEPTOR ANTAGONISTS JANSSEN PHARMACEUTICA NV (BE) 2010-04-22 WO disclosed