SCHEMBL3350867

SCHEMBL3350867

C[C@H](NC(=O)[C@@H]1CNC[C@H]1c1ccc(C(F)(F)F)nc1)c1cccc(Cl)c1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.52
ROCK2 O75116 2/20 0.39
MAPK1 P28482 4/20 0.39
TRPV1 Q8NER1 1/20 0.39
P2RX7 Q99572 2/20 0.38
KCNQ3 O43525 1/20 0.37
KCNQ2 O43526 1/20 0.37
KCNQ4 P56696 1/20 0.37
KCNQ5 Q9NR82 1/20 0.37
KIT P10721 2/20 0.36
TRPM8 Q7Z2W7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3347928 0.90 KCNH2 (0.53) KCNH2ROCK2MAPK1KCNQ3KCNQ2
SCHEMBL3348192 0.89 KCNH2 (0.57) KCNH2KCNQ3KCNQ2KCNQ4KCNQ5
SCHEMBL3348168 0.88 KCNH2 (0.45) KCNH2ROCK2MAPK1KCNQ3KCNQ2
SCHEMBL3346506 0.88 KCNH2 (0.51) KCNH2ROCK2
SCHEMBL3346354 0.86 KCNH2 (0.67) KCNH2ROCK2KCNQ3KCNQ2KCNQ4
SCHEMBL3353009 0.86 KCNH2 (0.67) KCNH2ROCK2KCNQ3KCNQ2KCNQ4
SCHEMBL3415190 0.84 KCNH2 (0.59) KCNH2ROCK2P2RX7
SCHEMBL3346383 0.82 KCNH2 (0.50) KCNH2ROCK2MAPK1KIT
SCHEMBL3346727 0.81 KCNH2 (0.53) KCNH2ROCK2TRPM8
SCHEMBL3353108 0.81 KCNH2 (0.46) KCNH2ROCK2MAPK1KCNQ3KCNQ2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed