SCHEMBL3348168

SCHEMBL3348168

C[C@H](NC(=O)[C@@H]1CNC[C@H]1c1ccc(Cl)nc1)c1cccc(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.45
ROCK2 O75116 3/20 0.42
MAPK1 P28482 9/20 0.40
CHRNA7 P36544 3/20 0.39
KIT P10721 1/20 0.39
MAPK3 P27361 1/20 0.38
PRKG1 Q13976 1/20 0.38
KCNQ3 O43525 2/20 0.38
KCNQ2 O43526 2/20 0.38
KCNQ4 P56696 1/20 0.38
KCNQ5 Q9NR82 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13365125 0.91 KCNH2 (0.44) KCNH2ROCK2CHRNA7PRKG1KCNQ3
SCHEMBL3353108 0.90 KCNH2 (0.46) KCNH2ROCK2MAPK1CHRNA7KIT
SCHEMBL13365073 0.90 KCNH2 (0.50) KCNH2ROCK2CHRNA7KCNQ3KCNQ2
SCHEMBL3352431 0.89 ROCK2 (0.52) KCNH2ROCK2CHRNA7PRKG1
SCHEMBL3350867 0.88 KCNH2 (0.52) KCNH2ROCK2MAPK1KITKCNQ3
SCHEMBL3353143 0.84 KCNH2 (0.53) KCNH2ROCK2CHRNA7KCNQ3KCNQ2
SCHEMBL3350804 0.83 MAPK1 (0.41) KCNH2ROCK2MAPK1KITMAPK3
SCHEMBL3346354 0.82 KCNH2 (0.67) KCNH2ROCK2KCNQ3KCNQ2KCNQ4
SCHEMBL3353009 0.82 KCNH2 (0.67) KCNH2ROCK2KCNQ3KCNQ2KCNQ4
SCHEMBL3413819 0.82 KCNH2 (0.42) KCNH2ROCK2MAPK1CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed