SCHEMBL3346727

SCHEMBL3346727

Cc1cccc([C@H](C)NC(=O)[C@@H]2CNC[C@H]2c2ccc(C(F)(F)F)nc2)n1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.53
HDAC4 P56524 1/20 0.37
TRPM8 Q7Z2W7 1/20 0.37
HRH3 Q9Y5N1 1/20 0.35
SSTR4 P31391 3/20 0.35
ROCK2 O75116 1/20 0.34
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34
ACACB O00763 1/20 0.34
ACKR3 P25106 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346260 0.89 KCNH2 (0.51) KCNH2HDAC4TRPM8HRH3ROCK2
SCHEMBL3346204 0.87 KCNH2 (0.54) KCNH2HDAC4TRPM8HRH3SSTR4
SCHEMBL3346658 0.86 KCNH2 (0.40) KCNH2SSTR4ROCK2
SCHEMBL3348192 0.84 KCNH2 (0.57) KCNH2HDAC4TRPM8ACACB
SCHEMBL3347928 0.82 KCNH2 (0.53) KCNH2HDAC4TRPM8ROCK2
SCHEMBL3353119 0.82 KCNH2 (0.47) KCNH2SSTR4PSEN1PSEN2APH1B
SCHEMBL3347822 0.82 KCNH2 (0.45) KCNH2ROCK2
SCHEMBL3345898 0.81 KCNH2 (0.54) KCNH2HDAC4TRPM8HRH3SSTR4
SCHEMBL3415190 0.81 KCNH2 (0.59) KCNH2HDAC4HRH3ROCK2ACACB
SCHEMBL3350867 0.81 KCNH2 (0.52) KCNH2TRPM8ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO claimed
WO-2010059922-A1 PYRROLIDINE CARBOXAMIDE COMPOUNDS LIGAND PHARMACEUTICALS INCORPORATED (US) 2010-05-27 WO disclosed