SCHEMBL3351783

SCHEMBL3351783

COc1ccc(COc2c(C(=O)O)cnc3ccc(=O)n(C)c23)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.44
POLB P06746 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ALKBH1 Q13686 1/20 0.42
PTPN1 P18031 1/20 0.41
PLA2G4B P0C869 1/20 0.40
FFAR1 O14842 5/20 0.40
KDM4E B2RXH2 1/20 0.39
ASPH Q12797 1/20 0.39
RIOX2 Q8IUF8 1/20 0.39
KDM8 Q8N371 1/20 0.39
PIK3CD O00329 1/20 0.39
MAOB P27338 1/20 0.39
KDM5A P29375 1/20 0.39
KDM4C Q9H3R0 1/20 0.39
KDM5B Q9UGL1 1/20 0.39
EGLN1 Q9GZT9 1/20 0.39
HDAC8 Q9BY41 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3346955 0.90 PLK1 (0.42) NPC1POLBRAB9ASMN1; SMN2ALKBH1
SCHEMBL3377466 0.90 MAOB (0.40) NPC1POLBRAB9ASMN1; SMN2ALKBH1
SCHEMBL3345433 0.81 CSF1R (0.41) KDM4EPIK3CD
SCHEMBL21679225 0.70 RAB9A (0.54) NPC1POLBRAB9ASMN1; SMN2ALKBH1
SCHEMBL9356673 0.70 RAB9A (0.56) NPC1POLBRAB9ASMN1; SMN2PLA2G4B
SCHEMBL691628 0.69 RAB9A (0.55) NPC1POLBRAB9ASMN1; SMN2PLA2G4B
SCHEMBL14699947 0.69 NPC1 (0.55) NPC1POLBRAB9ASMN1; SMN2PLA2G4B
SCHEMBL15680345 0.68 NPC1 (0.48) NPC1POLBRAB9ASMN1; SMN2ALKBH1
SCHEMBL14699822 0.68 SMN1; SMN2 (0.54) NPC1POLBRAB9ASMN1; SMN2PTPN1
SCHEMBL21179152 0.68 CYP1A2 (0.46) NPC1RAB9ASMN1; SMN2MAOBHDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010046388-A1 SUBSTITUTED (AZA) -1-METHYL-1H-QUINOLIN-2-ONES AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2010-04-29 WO disclosed
WO-2010045987-A1 SUBSTITUTED (AZA) -1-METHYL-1H-QUIN0LIN-2-0NES AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2010-04-29 WO disclosed