SCHEMBL3353828

SCHEMBL3353828

COCc1cccc(C#C[Si](C)(C)C)c1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.51
FFAR1 O14842 1/20 0.51
ERN1 O75460 1/20 0.35
IDO1 P14902 2/20 0.34
AGXT P21549 2/20 0.34
CYP2D6 P10635 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL510448 0.88 GRM5 (0.44) GRM5FFAR1IDO1AGXTCYP2D6
SCHEMBL15688010 0.84 TSHR (0.47) GRM5FFAR1CYP2D6HRH3MAOB
SCHEMBL22894412 0.81 FFAR1 (0.55) GRM5FFAR1ERN1IDO1AGXT
SCHEMBL2797815 0.81 GRM5 (0.38) GRM5IDO1CYP2D6HRH3
SCHEMBL3346401 0.80 ALDH1A1 (0.50) GRM5FFAR1MAOB
SCHEMBL24969103 0.79 GRM5 (0.38) GRM5CYP2D6HRH3
SCHEMBL3351697 0.79 FFAR1 (0.48) GRM5FFAR1CYP2D6HRH3
SCHEMBL18316997 0.79 FFAR1 (0.42) GRM5FFAR1MAOB
SCHEMBL19440746 0.78 CYP2D6 (0.39) GRM5FFAR1CYP2D6HRH3
SCHEMBL8850812 0.78 HRH3 (0.47) GRM5CYP2D6HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed