SCHEMBL3354058

SCHEMBL3354058

CCOC(=O)c1ccnc(C#C[Si](C)(C)C)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 1/20 0.50
JMJD6 Q6NYC1 4/20 0.49
CA12 O43570 3/20 0.44
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
CA7 P43166 3/20 0.44
CA9 Q16790 3/20 0.44
CA14 Q9ULX7 3/20 0.44
GABRA1 P14867 2/20 0.44
GABRA5 P31644 2/20 0.44
GABRG2 P18507 1/20 0.44
GABRB3 P28472 1/20 0.44
GABRA3 P34903 1/20 0.44
GABRA2 P47869 1/20 0.44
GABRA4 P48169 1/20 0.44
GABRA6 Q16445 1/20 0.44
KDM5A P29375 1/20 0.41
KDM5C P41229 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
KDM5B Q9UGL1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29851835 0.84 KDM4E (0.51) JMJD6CA12CA1CA2CA7
SCHEMBL1758901 0.84 KDM4E (0.51) JMJD6CA12CA1CA2CA7
SCHEMBL508971 0.81 JMJD6 (0.52) PIK3CAJMJD6CA12CA1CA2
SCHEMBL28940585 0.79 MEN1 (0.36) GABRA1GABRA5GABRG2GABRB3GABRA3
SCHEMBL2928318 0.79 CYP3A4 (0.50) CA12CA1CA2CA7CA9
SCHEMBL5680334 0.76 L3MBTL1 (0.46) PIK3CAJMJD6HSD17B2MEN1KMT2A
SCHEMBL3347534 0.76 JMJD6 (0.46) PIK3CAJMJD6MEN1NPC1RAB9A
SCHEMBL936599 0.76 ACACB (0.53) CA12CA1CA2CA7CA9
SCHEMBL363249 0.76 JMJD6 (0.58) PIK3CAJMJD6CA12CA1CA2
SCHEMBL30171421 0.76 JMJD6 (0.76) PIK3CAJMJD6CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed