SCHEMBL5680334

SCHEMBL5680334

CCOC(=O)c1ccnc(C#Cc2cc(OC)c(OC)c(OC)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.46
HSD17B2 P37059 1/20 0.46
JMJD6 Q6NYC1 3/20 0.43
BRAF P15056 1/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 2/20 0.42
CYP1A2 P05177 2/20 0.42
MAPT P10636 2/20 0.42
CYP1A1 P04798 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP1B1 Q16678 1/20 0.42
PIK3CA P42336 1/20 0.41
HPGD P15428 2/20 0.40
TSHR P16473 1/20 0.40
CYP3A4 P08684 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
PDGFRB P09619 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5679770 0.84 KDM4C (0.44) L3MBTL1KMT2AMEN1KDM4EALDH1A1
SCHEMBL4122249 0.78 JMJD6 (0.55) L3MBTL1HSD17B2JMJD6BRAFKMT2A
SCHEMBL3354058 0.76 PIK3CA (0.50) HSD17B2JMJD6KMT2AMEN1CYP1A2
SCHEMBL508971 0.74 JMJD6 (0.52) HSD17B2JMJD6KDM4EALDH1A1CYP1A2
Ethyltrimethoxy Benzoate SCHEMBL4410910 0.73 KMT2A (0.66) L3MBTL1HSD17B2KMT2AMEN1KDM4E
SCHEMBL5680000 0.73 GAA (0.39)
SCHEMBL7456502 0.71 JMJD6 (0.55) HSD17B2JMJD6CYP1A2PIK3CACYP3A4
SCHEMBL2765372 0.70 HPGD (0.61) KMT2AMEN1KDM4EALDH1A1CYP1A2
SCHEMBL3347534 0.70 JMJD6 (0.46) JMJD6KMT2AMEN1KDM4EALDH1A1
SCHEMBL3710171 0.70 KDM4E (0.52) L3MBTL1JMJD6KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1403249-B1 CYCLIC DIAMINE COMPOUNDS BEARING SIX-MEMBERED CYCLIC GROUPS KOWA CO (JP) 2006-03-15 EP disclosed
EP-1403249-A1 CYCLIC DIAMINE COMPOUNDS BEARING SIX-MEMBERED CYCLIC GROUPS Kowa Co., Ltd. (JP) 2004-03-31 EP disclosed
US-6509329-B1 Inhibitory effects on both cell adhesion and cell infiltration and is useful as a medicine for prevention or treatment of diseases such as allergy, asthma, rheumatism, arteriosclerosis and inflammation KOWA CO., LTD. (JP) 2003-01-21 US disclosed