SCHEMBL3354068

SCHEMBL3354068

CCOC(=O)c1ccncc1C#C[Si](C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.43
TSHR P16473 2/20 0.42
GABRA1 P14867 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
GABRA4 P48169 1/20 0.41
GABRA6 Q16445 1/20 0.41
TP53 P04637 1/20 0.41
CASP1 P29466 1/20 0.40
CDC7 O00311 1/20 0.40
DBF4 Q9UBU7 1/20 0.40
KDM5A P29375 1/20 0.39
KDM5B Q9UGL1 1/20 0.39
ALDH1A1 P00352 4/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31339220 0.82 TSHR (0.47) NUDT1TSHRTP53CASP1CDC7
SCHEMBL3515887 0.77 TSHR (0.60) NUDT1TSHRTP53CASP1CDC7
SCHEMBL29837473 0.77 TSHR (0.60) NUDT1TSHRTP53CASP1CDC7
SCHEMBL3290788 0.76 TSHR (0.50) NUDT1TSHRTP53CASP1CDC7
SCHEMBL277304 0.76 TSHR (0.53) NUDT1TSHRTP53CASP1CDC7
SCHEMBL31366358 0.75 TSHR (0.46) NUDT1TSHRTP53CASP1CDC7
SCHEMBL3879504 0.75 GABRA1 (0.47) TSHRGABRA1GABRG2GABRB3GABRA5
SCHEMBL3347544 0.75 OGA (0.40) NUDT1TSHRTP53ALDH1A1KMT2A
SCHEMBL13758656 0.74 TSHR (0.52) NUDT1TSHRTP53CASP1CDC7
SCHEMBL12447815 0.74 TSHR (0.52) NUDT1TSHRTP53CASP1CDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010063487-A1 PYRAZOLOPYRIMIDINES, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICINE MERZ PHARMA GMBH & CO. KGAA (DE) 2010-06-10 WO disclosed