Florbetapir F 18

Florbetapir F 18

SCHEMBL3356981

CNc1ccc(C=Cc2ccc(OCCOCCOCCF)nc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
APP P05067 20/20 1.00
MAPT P10636 1/20 1.00
SNCA P37840 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Florbetapir SCHEMBL29375540 1.00 APP (1.00) APPMAPTSNCA
Florbetapir SCHEMBL3356976 1.00 APP (1.00) APPMAPTSNCA
Florbetapir F 18 SCHEMBL14826096 1.00 APP (1.00) APPMAPTSNCA
Florbetapir F 18 SCHEMBL29517039 1.00 APP (1.00) APPMAPTSNCA
SCHEMBL13863151 0.92 APP (0.85) APPMAPTSNCA
SCHEMBL15307628 0.92 APP (0.85) APPMAPTSNCA
SCHEMBL15731546 0.90 APP (0.81) APPMAPTSNCA
SCHEMBL13827030 0.90 APP (0.81) APPMAPTSNCA
SCHEMBL12318871 0.90 APP (0.81) APPMAPTSNCA
SCHEMBL13827059 0.88 APP (0.79) APPMAPTSNCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 30 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2575898-B1 METHOD FOR PRODUCTION OF F-18 LABELED AMYLOID BETA LIGAND LIFE MOLECULAR IMAGING SA (CH) 2020-09-30 EP disclosed
EP-2579902-B2 METHOD FOR PRODUCTION OF F-18 LABELED AMYLOID BETA LIGANDS PIRAMAL IMAGING SA (CH) 2019-08-14 EP disclosed
EP-2590683-B1 METHOD FOR PRODUCTION OF F-18 LABELED AMYLOID BETA LIGANDS PIRAMAL IMAGING SA (CH) 2017-10-18 EP disclosed
EP-2579902-B1 METHOD FOR PRODUCTION OF F-18 LABELED AMYLOID BETA LIGANDS PIRAMAL IMAGING SA (CH) 2017-07-12 EP disclosed
EP-2363392-B1 STYRYLPYRIDINE DERIVATIVES AND THEIR USE FOR BINDING AND IMAGING AMYLOID PLAQUES UNIV PENNSYLVANIA (US) 2017-05-03 EP disclosed
US-9592308-B2 Method for production of F-18 labeled amyloid beta ligands PIRAMAL IMAGING SA (CH) 2017-03-14 US disclosed
US-20160184465-A1 METHOD FOR PRODUCTION OF F-18 LABELED AMYLOID BETA LIGANDS PIRAMAL IMAGING SA (CH) 2016-06-30 US disclosed
US-8981156-B2 Method for production of F-18 labeled amyloid beta ligands PIRAMAL IMAGING SA (CH) 2015-03-17 US disclosed
US-8840866-B2 Styrylpyridine derivatives and their use for binding and imaging amyloid plaques THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2014-09-23 US disclosed
US-20140243533-A1 METHOD FOR PRODUCTION OF F-18 LABELED A-BETA LIGANDS PIRAMAL IMAGING SA (CH) 2014-08-28 US disclosed
EP-2575898-A1 METHOD FOR PRODUCTION OF F-18 LABELED AMYLOID BETA LIGAND Piramal Imaging SA (CH) 2013-04-10 EP disclosed
EP-1999109-B1 STYRYLPYRIDINE DERIVATIVES AND THEIR USE FOR BINDING AND IMAGING AMYLOID PLAQUES UNIV PENNSYLVANIA (US) 2011-12-28 EP disclosed
WO-2011151273-A1 METHOD FOR PRODUCTION OF F-18 LABELED AMYLOID BETA LIGANDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-12-08 WO disclosed
WO-2011151282-A1 METHOD FOR PRODUCTION OF F-18 LABELED AMYLOID BETA LIGAND BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-12-08 WO disclosed
WO-2011151283-A1 METHOD FOR PRODUCTION OF F-18 LABELED AMYLOID BETA LIGANDS BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2011-12-08 WO disclosed
US-7687052-B2 radiolabeling; neurodegenerative diseases THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2010-03-30 US disclosed
US-20090123369-A1 Styrylpyridine Derivatives and Their Use for Binding and Imaging Amyloid Plaques THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2009-05-14 US disclosed
EP-1999109-A2 STYRYLPYRIDINE DERIVATIVES AND THEIR USE FOR BINDING AND IMAGING AMYLOID PLAQUES The Trustees Of The University Of Pennsylvania (US) 2008-12-10 EP disclosed
US-20080038195-A1 radiolabeling; neurodegenerative diseases THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2008-02-14 US disclosed
WO-2007126733-A2 STYRYLPYRIDINE DERIVATIVES AND THEIR USE FOR BINDING AND IMAGING AMYLOID PLAQUES THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2007-11-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160184465-A1 METHOD FOR PRODUCTION OF F-18 LABELED AMYLOID BETA LIGANDS APP, APBA1, BACE1 APP 1/4885MAPT 10/4885SNCA 9/4885
US-20140243533-A1 METHOD FOR PRODUCTION OF F-18 LABELED A-BETA LIGANDS FOLR2, FOLR1, ADRA2A APP 581/4885MAPT 2047/4885SNCA 232/4885
US-20080038195-A1 radiolabeling; neurodegenerative diseases APP, PSEN1, HTT APP 1/4885MAPT 6/4885SNCA 10/4885
US-20090123369-A1 Styrylpyridine Derivatives and Their Use for Binding and Imaging Amyloid Plaques APP, APBA1, PSEN1 APP 1/4885MAPT 7/4885SNCA 33/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.