SCHEMBL335772

SCHEMBL335772

CC(=O)NC(c1ccccc1F)[C@@H](O)C(=O)OC(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA7 P36544 1/20 0.37
CHRNA4 P43681 1/20 0.37
HTR3A P46098 1/20 0.37
CYP3A4 P08684 1/20 0.37
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
GAA P10253 1/20 0.37
LMNA P02545 2/20 0.36
ALDH1A1 P00352 1/20 0.36
CNR2 P34972 1/20 0.36
ROCK2 O75116 2/20 0.36
ROCK1 Q13464 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MC4R P32245 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL336016 0.84 CASP1 (0.39) GAALMNAALDH1A1L3MBTL1
SCHEMBL4102918 0.81 GAA (0.44) MEN1KMT2ACES2CES1GAA
SCHEMBL28573250 0.80 HTT (0.44) KMT2ACYP3A4GAAALDH1A1
SCHEMBL28573252 0.80 HTT (0.44) KMT2ACYP3A4GAAALDH1A1
SCHEMBL4178016 0.78 HTT (0.44) MEN1KMT2ACHRNB2CHRNB4CHRNA3
SCHEMBL19658634 0.73 L3MBTL1 (0.50) MEN1KMT2ACES2CES1GAA
SCHEMBL13050559 0.72 KMT2A (0.36) MEN1KMT2ACHRNB2CHRNB4CHRNA3
SCHEMBL13584745 0.71 ALDH1A1 (0.41) ALDH1A1L3MBTL1
SCHEMBL5021257 0.71 ALDH1A1 (0.41) ALDH1A1L3MBTL1
SCHEMBL4543253 0.71 ALDH1A1 (0.41) ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8097758-B2 Isoserine derivatives for use as coagulation factor IXa inhibitors SANOFI-AVENTIS (FR) 2012-01-17 US disclosed