SCHEMBL3358947

SCHEMBL3358947

COc1cc(-c2cc3c(c(Nc4ccc(N5CCOCC5)cc4)n2)C(=O)[N]C=C3)ncn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.40
MAPT P10636 4/20 0.39
MAPK1 P28482 2/20 0.39
HTT P42858 2/20 0.39
AHR P35869 1/20 0.39
ABL1 P00519 1/20 0.39
NTRK1 P04629 1/20 0.39
YES1 P07947 1/20 0.39
KDR P35968 1/20 0.39
PKMYT1 Q99640 1/20 0.39
TTBK1 Q5TCY1 1/20 0.39
TTBK2 Q6IQ55 1/20 0.39
ULK1 O75385 1/20 0.39
ZAP70 P43403 2/20 0.39
JAK2 O60674 3/20 0.38
JAK3 P52333 3/20 0.38
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
RAB9A P51151 1/20 0.38
EGFR P00533 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3362714 0.84 ABL1 (0.45) MAPTMAPK1ABL1NTRK1YES1
SCHEMBL3359607 0.84 KDR (0.41) MAPTMAPK1ABL1NTRK1YES1
SCHEMBL3360279 0.83 ABL1 (0.41) MAPTMAPK1ABL1NTRK1YES1
SCHEMBL3358758 0.81 SYK (0.44) MAPTMAPK1PKMYT1ZAP70JAK2
SCHEMBL3358312 0.81 MAPT (0.46) MAPTMAPK1ABL1KDRZAP70
SCHEMBL3359647 0.81 MAPT (0.43) MAPTMAPK1ZAP70TP53SYK
SCHEMBL3362709 0.81 SYK (0.45) MAPTMAPK1PKMYT1ZAP70TP53
SCHEMBL3362463 0.80 ZAP70 (0.49) MAPTMAPK1PKMYT1ZAP70JAK2
SCHEMBL3362540 0.80 SYK (0.44) MAPTMAPK1ABL1NTRK1YES1
SCHEMBL3358598 0.80 SYK (0.43) MAPTMAPK1ABL1KDRZAP70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2238137-A1 COMPOUNDS AND COMPOSITIONS AS KINASE INHIBITORS IRM LLC (BM) 2010-10-13 EP disclosed
WO-2009097287-A1 COMPOUNDS AND COMPOSITIONS AS KINASE INHIBITORS IRM LLC (BM) 2009-08-06 WO disclosed