SCHEMBL3360017

SCHEMBL3360017

Cc1c(O)c(=O)[nH]c2ccccc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 1.00
DDO Q99489 1/20 1.00
KDM4E B2RXH2 7/20 0.69
ALDH1A1 P00352 7/20 0.69
MAPT P10636 3/20 0.69
IDE P14735 1/20 0.69
MPI P34949 1/20 0.69
CACNA1B Q00975 1/20 0.69
APBA1 Q02410 1/20 0.69
RAB9A P51151 1/20 0.56
HPGD P15428 4/20 0.55
HSD17B10 Q99714 4/20 0.55
GRIN2D O15399 1/20 0.54
GRIN3B O60391 1/20 0.54
GRIN1 Q05586 1/20 0.54
GRIN2A Q12879 1/20 0.54
GRIN2B Q13224 1/20 0.54
GRIN2C Q14957 1/20 0.54
GRIN3A Q8TCU5 1/20 0.54
GAA P10253 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7807589 0.89 DAO (0.80) DAODDOKDM4EALDH1A1MAPT
SCHEMBL2726546 0.85 DAO (0.73) DAODDOKDM4EALDH1A1MAPT
SCHEMBL29505902 0.85 DAO (0.73) DAODDOKDM4EALDH1A1MAPT
SCHEMBL6220014 0.82 DAO (0.69) DAODDOKDM4EALDH1A1MAPT
SCHEMBL1884123 0.82 KDM4E (1.00) DAODDOKDM4EALDH1A1MAPT
SCHEMBL15690621 0.78 KDM4E (0.71) DAODDOKDM4EALDH1A1MAPT
SCHEMBL31182999 0.78 KDM4E (0.65) DAODDOKDM4EALDH1A1MAPT
SCHEMBL6923012 0.78 KDM4E (0.65) DAODDOKDM4EALDH1A1MAPT
SCHEMBL1276512 0.77 KDM4E (0.69) DAODDOKDM4EALDH1A1MAPT
SCHEMBL7567951 0.77 DAO (0.62) DAODDOKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9701638-B2 Therapeutic hydroxyquinolones RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2017-07-11 US disclosed
US-9701638-B2 Therapeutic hydroxyquinolones RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2017-07-11 US disclosed
US-9701638-B2 Therapeutic hydroxyquinolones RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2017-07-11 US disclosed
US-9468669-B2 Methods to treat dysregulated blood glucose disorders REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2016-10-18 US disclosed
US-9468669-B2 Methods to treat dysregulated blood glucose disorders REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2016-10-18 US disclosed
US-20160228515-A1 METHODS TO TREAT DYSREGULATED BLOOD GLUCOSE DISORDERS REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2016-08-11 US disclosed
US-20160228515-A1 METHODS TO TREAT DYSREGULATED BLOOD GLUCOSE DISORDERS REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2016-08-11 US disclosed
US-9339482-B2 Methods to treat dysregulated blood glucose disorders REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2016-05-17 US disclosed
US-9339482-B2 Methods to treat dysregulated blood glucose disorders REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2016-05-17 US disclosed
US-20150291531-A1 THERAPEUTIC HYDROXYQUINOLONES RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2015-10-15 US disclosed
US-20150291531-A1 THERAPEUTIC HYDROXYQUINOLONES RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2015-10-15 US disclosed
US-20150291531-A1 THERAPEUTIC HYDROXYQUINOLONES RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2015-10-15 US disclosed
US-20150150836-A1 METHODS TO TREAT DYSREGULATED BLOOD GLUCOSE DISORDERS REGENTS OF THE UNIVERSITY OF MINNESOTA 2015-06-04 US disclosed
US-20150150836-A1 METHODS TO TREAT DYSREGULATED BLOOD GLUCOSE DISORDERS REGENTS OF THE UNIVERSITY OF MINNESOTA 2015-06-04 US disclosed
WO-2014074926-A1 THERAPEUTIC HYDROXYQUINOLONES RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2014-05-15 WO disclosed
WO-2014074926-A1 THERAPEUTIC HYDROXYQUINOLONES RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2014-05-15 WO disclosed
WO-2010058314-A1 HYDROXYQUINOLIN-2(1H)-ONES AND DERIVATIVES THEREOF PFIZER INC. (US) 2010-05-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150291531-A1 THERAPEUTIC HYDROXYQUINOLONES RECQL, DDX5, DHX35 DAO 3157/4885DDO 3888/4885KDM4E 1278/4885
US-20150150836-A1 METHODS TO TREAT DYSREGULATED BLOOD GLUCOSE DISORDERS SLC2A4, SLC2A2, SLC2A3 DAO 3050/4885DDO 2128/4885KDM4E 3795/4885
US-20160228515-A1 METHODS TO TREAT DYSREGULATED BLOOD GLUCOSE DISORDERS SLC2A4, SLC2A2, SLC2A3 DAO 3050/4885DDO 2128/4885KDM4E 3795/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.