SCHEMBL3360283

SCHEMBL3360283

CCCCc1ncccc1SSc1cccnc1CCCN

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.40
HRH1 P35367 6/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
CASP3 P42574 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
TLR8 Q9NR97 1/20 0.33
CXCR4 P61073 4/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP19A1 P11511 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3082743 0.89 HRH1 (0.46) CYP2A6HRH1CXCR4CHRNA7
SCHEMBL13095176 0.81 HRH1 (0.44) CYP2A6HRH1L3MBTL1TDP1ALDH1A1
SCHEMBL3081098 0.78 CYP2A6 (0.40) CYP2A6HRH1CXCR4HTR2ACHRNA7
SCHEMBL8735931 0.75 TLR8 (0.47) CYP2A6HRH1L3MBTL1TDP1TLR8
SCHEMBL13095210 0.74 ALDH1A1 (0.38) HRH1L3MBTL1TDP1ALDH1A1HPGD
SCHEMBL253769 0.73 L3MBTL1 (0.40) CYP2A6L3MBTL1TDP1NPC1ALDH1A1
Phosphoric Acid SCHEMBL28641959 0.73 PDE3B (0.35) L3MBTL1ALDH1A1HPGDSMN1; SMN2
SCHEMBL19865639 0.73 L3MBTL1 (0.42) L3MBTL1TDP1NPC1ALDH1A1HPGD
SCHEMBL510211 0.73 CYP2C9 (0.43) L3MBTL1TDP1HPGDTLR8CXCR4
SCHEMBL8764979 0.73 L3MBTL1 (0.42) L3MBTL1TDP1NPC1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2205600-A1 CARBACEPHEM ß -LACTAM ANTIBIOTICS Achaogen, Inc. (US) 2010-07-14 EP disclosed
WO-2010030811-A2 CARBACEPHEM β-LACTAM ANTIBIOTICS ACHAOGEN, INC. (US) 2010-03-18 WO disclosed
WO-2009055696-A1 CARBACEPHEM β-LACTAM ANTIBIOTICS ACHAOGEN, INC. (US) 2009-04-30 WO disclosed