SCHEMBL3362516

SCHEMBL3362516

COc1ncc(-c2cc3c(c(Nc4ccc(N5CCO[C@H](C)C5)c(F)c4)n2)C(=O)[N]C=C3)cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ZAP70 P43403 1/20 0.47
SYK P43405 3/20 0.35
BTK Q06187 2/20 0.35
EGFR P00533 1/20 0.35
P2RX3 P56373 2/20 0.34
JAK3 P52333 2/20 0.34
LCK P06239 1/20 0.34
MTOR P42345 2/20 0.34
SMO Q99835 1/20 0.34
LRRK2 Q5S007 1/20 0.33
PIK3CG P48736 2/20 0.33
PIK3CD O00329 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
CDK4 P11802 2/20 0.32
CSF1R P07333 1/20 0.32
CDK6 Q00534 1/20 0.32
CDK1 P06493 1/20 0.32
CCNB1 P14635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3362713 0.92 ZAP70 (0.56) ZAP70SYKP2RX3JAK3MTOR
SCHEMBL3359505 0.91 ZAP70 (0.47) ZAP70SYKBTKEGFRJAK3
SCHEMBL3362937 0.90 ZAP70 (0.48) ZAP70SYKBTKEGFRJAK3
SCHEMBL3358405 0.90 ZAP70 (0.46) ZAP70SYKBTKEGFRP2RX3
SCHEMBL3356910 0.90 MTOR (0.42) SYKBTKEGFRP2RX3JAK3
SCHEMBL3359492 0.89 ZAP70 (0.46) ZAP70SYKBTKEGFRJAK3
SCHEMBL3357809 0.88 SYK (0.44) ZAP70SYKBTKJAK3MTOR
SCHEMBL3362890 0.86 ZAP70 (0.39) ZAP70SYKBTKEGFRP2RX3
SCHEMBL3358595 0.86 ZAP70 (0.38) ZAP70SYKBTKEGFRP2RX3
SCHEMBL3357730 0.85 ZAP70 (0.55) ZAP70SYKP2RX3JAK3SMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2238137-A1 COMPOUNDS AND COMPOSITIONS AS KINASE INHIBITORS IRM LLC (BM) 2010-10-13 EP claimed
WO-2009097287-A1 COMPOUNDS AND COMPOSITIONS AS KINASE INHIBITORS IRM LLC (BM) 2009-08-06 WO claimed