SCHEMBL3363485

SCHEMBL3363485

Nc1cccc(-c2ccccc2Cl)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.58
MAOA P21397 1/20 0.56
MAP4K4 O95819 2/20 0.52
PLA2G7 Q13093 1/20 0.52
BACE1 P56817 1/20 0.49
JAK2 O60674 1/20 0.47
JAK1 P23458 1/20 0.47
TYK2 P29597 1/20 0.47
JAK3 P52333 1/20 0.47
ALDH1A1 P00352 2/20 0.46
SCN9A Q15858 1/20 0.45
CYP3A4 P08684 1/20 0.44
CASP1 P29466 1/20 0.44
RECQL P46063 1/20 0.44
MAPT P10636 3/20 0.44
BRD4 O60885 1/20 0.44
MAOB P27338 1/20 0.43
MECP2 P51608 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8307816 0.86 MAP4K4 (0.50) CYP2A6MAOAMAP4K4PLA2G7ALDH1A1
SCHEMBL29628996 0.84 CYP2A6 (0.71) CYP2A6BACE1JAK2JAK1TYK2
SCHEMBL9479255 0.84 CYP2A6 (0.71) CYP2A6BACE1JAK2JAK1TYK2
SCHEMBL29471388 0.84 MAOA (0.68) MAOAMAP4K4ALDH1A1CYP3A4CASP1
SCHEMBL2023695 0.84 MAOA (0.68) MAOAMAP4K4ALDH1A1CYP3A4CASP1
SCHEMBL2442271 0.82 MAOA (0.65) MAOAMAP4K4ALDH1A1CYP3A4CASP1
SCHEMBL7642404 0.80 MAOA (0.70) MAOAMAP4K4ALDH1A1CYP3A4CASP1
SCHEMBL30449021 0.80 MAOA (0.70) MAOAMAP4K4ALDH1A1CYP3A4CASP1
Ethane SCHEMBL28326570 0.80 MAOA (0.62) MAOAMAP4K4ALDH1A1CYP3A4CASP1
SCHEMBL29726725 0.80 MAOA (0.70) MAOAMAP4K4ALDH1A1CYP3A4CASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108440414-B Pyrazolone amide antifungal drug and preparation method and application thereof 中国人民解放军第二军医大学 2021-07-09 CN disclosed
CN-105985248-B A kind of method of synthesizing amino Diaromatic compound 上海泰禾国际贸易有限公司 2018-10-26 CN disclosed
EP-1984331-B1 PYRROLIDINE DERIVATIVES AS ERK INHIBITORS SCHERING CORP (US) 2010-10-20 EP disclosed
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed
WO-2010046780-A2 ANTI VIRAL COMPOUNDS INSTITUT PASTEUR KOREA (KR) 2010-04-29 WO disclosed
US-20040259875-A1 Amine derivatives BAYER HEALTHCARE AG (DE) 2004-12-23 US disclosed
EP-1414788-A1 NAPHTHYLUREA AND NAPHTHYLACETAMIDE DERIVATIVES AS VANILLOID RECEPTOR 1 (VR1) ANTAGONISTS Bayer HealthCare AG (DE) 2004-05-06 EP disclosed
WO-2003014064-A1 NAPHTHYLUREA AND NAPHTHYLACETAMIDE DERIVATIVES AS VANILLOID RECEPTOR 1 (VR1) ANTAGONISTS BAYER HEALTHCARE AG (DE) 2003-02-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040259875-A1 Amine derivatives AVPR1A, GRIN1, OPRL1 CYP2A6 4361/4885MAOA 1047/4885MAP4K4 1377/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.