SCHEMBL3363987

SCHEMBL3363987

COc1cc(OC)c2c(CNC(=O)OC(C)(C)C)ncc(C(=O)N(C)Cc3cccnc3)c2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 1/20 0.42
CYP3A4 P08684 3/20 0.40
TLR9 Q9NR96 1/20 0.39
TLR8 Q9NR97 1/20 0.39
TLR7 Q9NYK1 1/20 0.39
RECQL P46063 1/20 0.39
DPP4 P27487 2/20 0.39
PDK1 Q15118 3/20 0.39
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
NAMPT P43490 2/20 0.39
IDO1 P14902 1/20 0.38
CYP1A2 P05177 2/20 0.38
TSHR P16473 1/20 0.38
BLM P54132 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
RIPK1 Q13546 1/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3365615 0.92 DPP4 (0.41) DPP4GAAHTTMEN1KMT2A
SCHEMBL3361319 0.88 GAA (0.44) CLK1CYP3A4RECQLGAAHTT
SCHEMBL3363205 0.84 DPP4 (0.56) CLK1TLR9TLR8TLR7RECQL
Hydrochloric Acid SCHEMBL3366027 0.83 DPP4 (0.56) CLK1TLR9TLR8TLR7RECQL
SCHEMBL3363213 0.82 TLR8 (0.40) TLR9TLR8TLR7DPP4GAA
SCHEMBL3361777 0.82 TP53 (0.41) DPP4TSHRMEN1KMT2AMAPT
SCHEMBL3363088 0.80 DPP4 (0.41) DPP4MEN1KMT2AMAPTL3MBTL1
SCHEMBL3363099 0.79 DPP4 (0.49) DPP4GAACYP1A2TSHRSMN1; SMN2
SCHEMBL7716634 0.79 ABCC1 (0.38) DPP4GAAHTTTSHRMEN1
SCHEMBL3361175 0.79 HPGD (0.44) DPP4GAAHTTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed