SCHEMBL7716634

SCHEMBL7716634

COc1cc(OC)c2c(CNC(=O)OC(C)(C)C)ncc(NC(=O)N(C)Cc3ccccc3)c2c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 1/20 0.38
CTSL P07711 1/20 0.37
CTSB P07858 1/20 0.37
CTSS P25774 1/20 0.37
CKS1B P61024 1/20 0.37
SKP1 P63208 1/20 0.37
SKP2 Q13309 1/20 0.37
PTPN1 P18031 1/20 0.37
HTT P42858 3/20 0.36
TSHR P16473 2/20 0.36
ALOX15 P16050 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GAA P10253 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
NT5E P21589 1/20 0.35
ROCK2 O75116 1/20 0.35
CYP2C9 P11712 1/20 0.35
ROCK1 Q13464 1/20 0.35
CDC42BPA Q5VT25 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3361319 0.92 GAA (0.44) HTTSMN1; SMN2GAAMEN1KMT2A
SCHEMBL3366103 0.91 TSHR (0.40) CTSLCTSBCTSSPTPN1HTT
SCHEMBL3362011 0.88 DPP4 (0.40) CTSLCKS1BSKP1SKP2TSHR
SCHEMBL3361886 0.88 DPP4 (0.41) ABCC1CTSLCTSBCTSSCKS1B
SCHEMBL3365615 0.87 DPP4 (0.41) CTSLCTSBCTSSPTPN1HTT
SCHEMBL7720962 0.85 DPP4 (0.49) ABCC1HTTTSHRALOX15SMN1; SMN2
SCHEMBL7723483 0.83 GAA (0.40) HTTTSHRSMN1; SMN2GAAMEN1
SCHEMBL3361777 0.80 TP53 (0.41) CKS1BSKP1SKP2TSHRMEN1
SCHEMBL3360962 0.80 DPP4 (0.41) GAAKMT2ADPP4
SCHEMBL3363987 0.79 CLK1 (0.42) HTTTSHRSMN1; SMN2GAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed