SCHEMBL3365064

SCHEMBL3365064

COc1cc2c(CC(=O)N(C)CCc3ccccn3)cnc(CNC(=O)OC(C)(C)C)c2cc1OC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.43
ALDH1A1 P00352 3/20 0.43
TDP1 Q9NUW8 2/20 0.43
AVPR1B P47901 1/20 0.41
HIF1A Q16665 1/20 0.40
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TLR8 Q9NR97 2/20 0.38
TLR7 Q9NYK1 2/20 0.38
TLR9 Q9NR96 1/20 0.38
DPP4 P27487 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ATM Q13315 1/20 0.37
PDE10A Q9Y233 1/20 0.37
LTB4R Q15722 1/20 0.36
LTB4R2 Q9NPC1 1/20 0.36
RAF1 P04049 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3361800 0.84 CTSL (0.43) KMT2AMEN1DPP4LTB4RLTB4R2
SCHEMBL3363381 0.84 DPP4 (0.55) KDM4EALDH1A1TDP1AVPR1BHIF1A
Hydrochloric Acid SCHEMBL3369641 0.83 DPP4 (0.56) KDM4EALDH1A1TDP1AVPR1BHIF1A
SCHEMBL3363192 0.81 CYP3A4 (0.41) KDM4EALDH1A1KMT2AMEN1CYP1A2
SCHEMBL3362959 0.80 DPP4 (0.40) DPP4PDE10A
SCHEMBL3360434 0.78 DPP4 (0.41) ALDH1A1KMT2AMEN1DPP4PDE10A
SCHEMBL3361880 0.78 DPP4 (0.47) DPP4PDE10A
SCHEMBL3362196 0.78 DPP4 (0.46) DPP4PDE10A
SCHEMBL3363213 0.77 TLR8 (0.40) KDM4EALDH1A1TDP1HIF1AKMT2A
SCHEMBL3362189 0.74 DPP4 (0.43) KDM4ECYP1A2DPP4ATMPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7732446-B1 Dipeptidyl peptidase inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-06-08 US disclosed